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(4aS,7aR)-1-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{[2-(2-hydroxyethyl)piperidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-{7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-3-(2,6-dimethylphenoxy)azetidine
1-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
(3S,4R)-1-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-4-(hydroxymethyl)piperidin-3-ol
[2,2-dimethyl-3-(morpholin-4-yl)propyl](methyl)[(1-methylpiperidin-3-yl)methyl]amine
1-[(2-methoxyphenyl)methyl]-3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidine
2-(oxan-2-ylmethoxy)-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
2-{[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-(4-fluorophenyl)-1-(5-hydroxypyrazine-2-carbonyl)piperazine-2-carboxamide
1-(cyclohexylmethyl)-3-hydroxy-3-{[(pyridin-3-ylmethyl)amino]methyl}piperidin-2-one
N-{1-[1-(2,3-difluorobenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylthiophene-3-carboxamide
7-[3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-cyclopentyl-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N-cyclopentyl-3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
2-{[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]methyl}-6-methyl-4-(thiomorpholin-4-yl)quinazoline
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
1-(3,5-dimethylphenyl)-4-[2-(pyrrolidin-1-yl)benzoyl]piperazin-2-one
6-(4-methoxyphenyl)-N-methyl-8-oxo-7-(prop-2-en-1-yl)-N-(propan-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(7R,9aR)-7-[(benzylsulfanyl)methyl]-6,9-dioxo-N-phenyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
1-benzyl-4-oxo-N3-(prop-2-en-1-yl)-N5-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(3S)-1-ethyl-3-methyl-4-{[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperazin-2-one
5-(propan-2-yl)-N-[2-(1H-1,2,4-triazol-1-yl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3,5-difluoro-N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]pyridine-2-carboxamide
6-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)pyridine-2-carbonitrile
3-(pyridin-4-yl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-1H-pyrazole-5-carboxamide
4-ethyl-5-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]-1,3-thiazol-2-amine
2-fluoro-6-methoxy-4-({8-methyl-2,8-diazaspiro[4.5]decan-2-yl}methyl)phenol
N-(2-methanesulfonamidoethyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
N-(3-phenylpropyl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
methyl({[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl})[1-(pyrimidin-4-yl)ethyl]amine
(3S,4R)-4-(2-methylphenyl)-1-(pyrimidin-5-ylmethyl)pyrrolidine-3-carboxylic acid
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-methoxypyrimidine-5-carboxamide
4-[(1H-imidazol-2-ylmethyl)amino]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}({[1-(pyrimidin-2-yl)piperidin-3-yl]methyl})amine
1-phenyl-N-(piperidin-4-yl)-N-(pyridin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
8-chloro-2-{[2-(2-methoxyethyl)morpholin-4-yl]methyl}quinoline
8-(5-chloro-2-hydroxybenzoyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
1-[(4-methoxyphenyl)methyl]-4-[2-(1-methyl-3-oxopiperazin-2-yl)acetyl]piperazin-2-one
6-[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
4-(thiomorpholin-4-yl)-N-[2-(trifluoromethyl)phenyl]piperidine-1-carboxamide
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-2-ethyl-4-methyl-1,3-thiazole-5-carboxamide
3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-{4-[(2-methylprop-2-en-1-yl)oxy]phenyl}-3-(propan-2-yl)urea
1-{2-[(benzylsulfamoyl)amino]ethyl}imidazolidin-2-one
(4aS,8aR)-6-(pyrazin-2-yl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,3,5-trimethyl-1,2-oxazole-4-carboxamide
1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide