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{4-[(2-chloro-5-methoxy-4-propoxyphenyl)methyl]morpholin-3-yl}methanol
N-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
4-[1-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carbonyl]morpholine
3-{[2-(dimethylsulfamoyl)ethyl]sulfamoyl}-N-(2-fluoroethyl)benzamide
ethyl[(5-propyl-1,2,4-oxadiazol-3-yl)methyl](quinoxalin-2-ylmethyl)amine
6-{7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-N-methylpyridine-2-carboxamide
{1-[4-(4-{[(1-phenylcyclopentyl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-yl}methanol
N-(2-oxopiperidin-3-yl)-4-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
[3-({1-[1-(pyridine-4-carbonyl)piperidin-4-yl]pyrrolidin-3-yl}methyl)phenyl]methanol
3-butanamido-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]benzamide
4-(3-phenyl-1,2,4-oxadiazol-5-yl)benzene-1-sulfonamide
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3,3,3-trifluoropropan-1-one
1-methyl-3-(2-methylpropyl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
methyl 3-(cyclobutylmethoxy)-5-{[(4-hydroxyphenyl)methyl]carbamoyl}benzoate
1,3-dimethyl-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-(3,4-diethoxybenzoyl)-3,9-diazaspiro[5.6]dodecan-10-one
N,N,5-trimethyl-2-(3-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidin-4-amine
methyl 5-[(4-hydroxy-4-methylpentan-2-yl)amino]-3-(2-methoxyacetamido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
N-(1H-indol-5-ylmethyl)-N-[(2-methoxyphenyl)methyl]cyclopropanamine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(1H-imidazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5,7-dimethyl-3-{2-oxo-2-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}-2,3-dihydro-1H-indol-2-one
8-chloro-2-ethyl-4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1-methylpiperidine-3-carboxamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-(1,2-oxazolidin-2-ylmethyl)piperidin-2-one
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidine-3-carboxylic acid
1-(cyclohex-3-en-1-ylmethyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-1H-pyrazole-3-carboxamide
1-[3-(2-fluorophenyl)-1H-pyrazole-4-carbonyl]-2-(furan-2-yl)azepane
N-{1-[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}pyrimidin-2-amine
diethyl[(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)sulfamoyl]amine
2-(3-methoxypropanamido)-N-[(3-methylphenyl)methyl]benzamide
N-methyl-2-(4-phenylpiperidin-1-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
2-{[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidin-1-yl]methyl}benzonitrile
4-(6-methyl-1H-1,3-benzodiazol-2-yl)-2,1,3-benzothiadiazole
2-(3-fluorophenyl)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
methyl (2S,4R)-1-[(4-methoxyphenyl)methyl]-4-(4-phenylbenzamido)pyrrolidine-2-carboxylate
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)pyrimidin-2-amine
N-methyl-2-[1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl]acetamide
methyl 5-[(4-ethoxyphenyl)carbamoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
5-ethyl-6-methyl-N4-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}pyrimidine-2,4-diamine
2-methoxy-3-{5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}quinoline
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-{spiro[azepane-4,2'-chromene]-1-yl}propan-1-one
6-(propan-2-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-4-amine
3-[5-(1-benzofuran-5-yl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
6-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}pyridine-2-carboxylic acid
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]acetamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-methanesulfonylpyrrolidine-3-carboxylic acid
2-(1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-4-yl)ethan-1-ol