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8-(2-chloro-4-fluorobenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-ethyl-3-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-5-(piperidin-4-yl)imidazolidine-2,4-dione
3-(4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperazin-1-yl)-1,2-benzothiazole
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
N-{[1-(2-hydroxybutyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
6-(2-aminoethyl)-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methylpyrimidin-4-amine
N-(2-hydroxyethyl)-3-(1-methylpiperidin-2-yl)-N-{[4-(methylsulfanyl)phenyl]methyl}propanamide
2-{5-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
7-methoxy-3-[6-(morpholine-4-carbonyl)pyrazin-2-yl]-2,3,4,5-tetrahydro-1H-3-benzazepine
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]pyrrolidin-3-yl]methanol
3-{[(2R)-2-methylpiperazin-1-yl]sulfonyl}-N-(thiophen-3-ylmethyl)benzamide
ethyl 4-[(2-chlorophenyl)methyl]-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidine-4-carboxylate
2-[(4-benzylpiperazin-1-yl)methyl]-1,3-oxazole-4-carboxylic acid
2-(4-{[5-(methoxymethyl)furan-2-yl]methyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-yl)ethan-1-ol
ethyl 1-benzyl-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-(4-methoxy-2-methylphenyl)-2-methyl-1H-imidazole
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-5-(methoxymethyl)-N-methylthiophene-2-carboxamide
3-cyclopropyl-1-(2,3-dimethylphenyl)-5-(1H-1,2,3-triazol-1-ylmethyl)-1H-1,2,4-triazole
6-(1-phenylcyclohexanecarbonyl)-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
5-[1-(2,4-difluorophenoxy)ethyl]-1-ethyl-3-(2-methoxyethyl)-1H-1,2,4-triazole
(3S,4S)-1-[3-(methylsulfanyl)propyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
4-[2-(2-methyl-1H-indol-3-yl)acetyl]-1-(2-methylphenyl)piperazin-2-one
4-ethyl-3-{[1-(2-ethylpyrimidine-5-carbonyl)piperidin-4-yl]methyl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-3-(methoxymethyl)pyrrolidine
1-(4-methyl-1,2,5-oxadiazol-3-yl)-4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperazine
6-cyclobutyl-1-[(4-methoxyphenyl)methyl]-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-(3-methylbutyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(4-methylphenyl)piperazine
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-1-methylpiperidine-3-carboxamide
1-cyclobutanecarbonyl-4-(3-phenylpropyl)piperidine-4-carboxylic acid
4-[5-(furan-3-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]-1H-pyrazole
3-(2-fluorophenyl)-6-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-hexanoylpyrrolidine-3-carboxylic acid
2-[4-(4-methoxyphenyl)-3,5-dimethyl-1H-pyrazol-1-yl]-N-(1-methyl-1H-indazol-3-yl)acetamide
N-{1-[4-(morpholine-4-carbonyl)pyridin-2-yl]piperidin-4-yl}methanesulfonamide
N-cyclopropyl-1-[1-(quinolin-5-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
N-[(5-chlorothiophen-2-yl)methyl]-1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
N-[(2-fluorophenyl)methyl]-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(1-{[5-(2-chlorophenyl)furan-2-yl]methyl}piperidin-4-yl)-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
2,3,5-trimethyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1-(furan-2-ylmethyl)piperidine
(1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-3-[(4-fluorophenyl)methyl]piperidin-3-yl)methanol
9-(4-methylbenzoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-3-yl]-3,5-dimethyl-1H-pyrazole
(3S)-N-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-amine
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-(2,5-dimethylphenyl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-{4-[(2-fluoro-5-methoxyphenyl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
N-{1-[1-(pyrimidin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
2-{2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenoxy}-N-methylacetamide