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1-(6-methyl-2-propylpyrimidin-4-yl)-N-[1-(pyrimidin-4-yl)ethyl]piperidin-4-amine
(2R,6R)-4-[(furan-2-ylmethyl)carbamoyl]-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]acetamide
3-[(3R,4S)-1-(1-benzothiophen-2-ylmethyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-2-(phenylsulfanyl)acetamide
4-[3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)propanoyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-(3-methoxybenzoyl)-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazine
N-benzyl-4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
2-cyclopropyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-(furan-2-ylmethyl)-2-(2-methyl-1,3-thiazol-4-yl)-N-(pyridin-2-ylmethyl)acetamide
2-(2,6-dimethoxypyridin-3-yl)-2-[4-(pyrrolidin-1-yl)piperidin-1-yl]acetic acid
3-(3,6-dimethylpyrazin-2-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
9-[2-(3-chlorophenyl)acetyl]-4-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
2-(2,3-dihydro-1H-inden-1-yl)-N-[1-(oxan-4-yl)piperidin-4-yl]acetamide
(3S,4S)-1-(3-methoxypyrazin-2-yl)-4-(naphthalen-2-yl)piperidin-3-ol
2,6-dimethyl-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]quinoline-4-carboxamide
4-[(1-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one
2-(3-chloro-4-hydroxyphenyl)-N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)acetamide
5-hydroxy-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]pyrazine-2-carboxamide
2-{[benzyl(3-hydroxy-2-methylpropyl)amino]methyl}-4-fluorophenol
3-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]benzene-1,2-diol
7-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4,5-dimethyl-6-[4-(1H-pyrazol-5-yl)phenyl]pyrimidine
5-cyclopropyl-N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-1,2-oxazole-3-carboxamide
({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)(pyridin-2-ylmethyl)amine
3-methyl-1-[1-(6-{[(5-methylfuran-2-yl)methyl]amino}pyridine-3-carbonyl)piperidin-3-yl]butan-1-one
3-fluoro-N-[2-(1H-indol-1-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
2-(propan-2-yl)-5-{1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-imidazol-2-yl}pyrimidine
3-cyclopropyl-1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
(3S)-3-ethyl-4-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]morpholine
7-(2-methyl-1,8-naphthyridine-3-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
ethyl({[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})(2-methylprop-2-en-1-yl)amine
(2S,3R)-2-amino-3-methyl-1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pentan-1-one
8-{5-[ethyl(methyl)carbamoyl]pyridin-2-yl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(pyridin-4-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]propanamide
4-methyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}pyrimidine-5-carboxamide
2-(3-methoxyphenyl)-7-phenyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-ethyl-N4-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrimidine-2,4-diamine
2-benzyl-N-(3-fluorophenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-[2-(2-oxopiperidin-1-yl)ethyl]piperidine-4-carboxamide
N-(1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
4-(2,3-dichlorophenyl)-3-[(methylamino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
[(3R,4S)-4-(morpholin-4-ylmethyl)-1-(3-phenylpropyl)pyrrolidin-3-yl]methanol
3-{[4-phenyl-5-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}pyridine
1-{2-[1-benzyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}piperidin-2-one
ethyl 4-[(4-chlorophenyl)methyl]-1-(1H-imidazol-2-ylmethyl)piperidine-4-carboxylate
4-benzyl-3-(piperidin-4-yl)-1-[2-(1H-pyrrol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-acetyl-N-{1-azabicyclo[2.2.2]octan-3-yl}-2,4-dimethyl-1H-pyrrole-3-carboxamide