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1-[4-(4-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-cyclohexylethan-1-one
1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(1H-pyrazol-1-ylmethyl)piperidine
1-(1-{[4-(dimethylamino)phenyl]methyl}piperidin-3-yl)-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl}){[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-1,3-oxazole-5-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]ethan-1-one
2-{2-[(3-ethylmorpholin-4-yl)methyl]phenyl}-3H,4H,5H,6H,7H,8H,9H-cyclohepta[d]pyrimidin-4-one
N-(2-{4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)-3-methylbenzamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}propanamide
6-(2,5-dimethylfuran-3-yl)-2-[(3S)-3-hydroxypyrrolidine-1-carbonyl]-7-(3-methylbut-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-cyclopropyl-1,4,6-trimethyl-N-[(3-methylthiophen-2-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(3S,4R)-1-(2,5-dimethylfuran-3-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2,3-dimethyl-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}quinoxaline-6-carboxamide
1,3,7-trimethyl-N-[2-(2-methylpropanesulfonyl)ethyl]-1H-indole-2-carboxamide
3-(cyclopentylsulfamoyl)-5-(2-methyl-1H-imidazol-1-yl)benzoic acid
2-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,3-benzothiazole
3-fluoro-5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]benzonitrile
1-(4-aminobutanoyl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-(4-fluorophenoxy)-N-(3,4,5-trimethoxyphenyl)azetidine-1-carboxamide
4-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-pyrazole
methyl({5-[(4-methyl-1H-imidazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)[2-(phenylsulfanyl)ethyl]amine
N-(1,4-dioxan-2-ylmethyl)-3,5-difluoropyridine-2-carboxamide
1-[(3ar,6ar)-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
2-benzyl-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-1,3-benzoxazole-5-carboxamide
6-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-2-carbonitrile
methyl[(1-{[1-(thiophen-2-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]amine
1-(4-methoxyphenyl)-N-methyl-N-[1-(pyridin-4-yl)ethyl]piperidin-4-amine
1-phenyl-4-(quinoxaline-6-carbonyl)piperazin-2-one
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-[2-(pyridin-3-ylformamido)ethyl]propanamide
4-cyclopropanecarbonyl-5-methyl-1-(4-methylphenyl)piperazin-2-one
1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
2-ethyl-4-({2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}methyl)pyrimidine
4-{3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-methyl-6-(1H-pyrazol-1-yl)pyrimidine
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]acetamide
[1-(furan-2-yl)ethyl]({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)methylamine
{3-[(4-fluorophenyl)methyl]-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidin-3-yl}methanol
2-[(1R,3S,3aS,6aR)-1-(hydroxymethyl)-5-methyl-3-[3-(2-methylpropoxy)phenyl]-octahydropyrrolo[3,4-c]pyrrol-1-yl]ethan-1-ol
4-benzyl-3-ethyl-1-[2-(ethylsulfanyl)ethyl]-1,4-diazepan-5-one
(4aS,8aR)-6-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
1-(4-hydroxyphenyl)-5-oxo-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)pyrrolidine-3-carboxamide
(1S,5R)-3-(4,6-dimethoxypyrimidin-2-yl)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(4-methoxy-2-methylphenyl)-3-(morpholin-4-yl)piperidine-1-carboxamide
methyl(pyridin-3-ylmethyl){[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}amine
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(4aR,8aS)-1-[(4-fluorophenyl)methyl]-6-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(3-chloro-2,6-difluorophenyl)ethan-1-one
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-(pyridin-4-yl)-1,4-diazepan-6-ol
1-benzyl-8-{[3-(furan-2-yl)phenyl]methyl}-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 4-{2-[(propan-2-yl)amino]pyrimidine-5-carbonyl}piperazine-1-carboxylate