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2,4-dichloro-6-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenol
2-[({1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]-N,N-dimethylacetamide
3-butyl-4-ethyl-1-(2-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-2-oxoethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-4-(4-{[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}phenyl)butan-2-ol
1-(1H-indol-2-ylmethyl)-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
2-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-5-methylpyrazine
7-(9H-fluoren-2-ylmethyl)-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,3-benzothiazole-6-carboxamide
2-(5-methyl-3-phenyl-1,2-oxazol-4-yl)-2-(morpholin-4-yl)acetic acid
8-[2-(3,4-dimethylphenyl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-({[1-(pyridin-4-ylmethyl)piperidin-3-yl]oxy}methyl)pyridine
4-[(2,5-dimethoxyphenyl)methyl]-9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N,N-diethyl-2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]acetamide
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(furan-2-ylmethyl)methylamine
2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)-N-(pyrimidin-4-ylmethyl)acetamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
N-({1-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
N-{1-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-2-phenylethyl}-2-(dimethylamino)-N-methylacetamide
1-methyl-4-[4-(1-methyl-1H-1,2,4-triazol-5-yl)phenyl]piperazine
methyl 5-{[(3,4-dimethoxyphenyl)methyl]amino}-3-(furan-3-amido)-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(3-chloro-4-methoxybenzenesulfonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-cyclohexyl-6-hydroxy-4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1,4-diazepan-2-one
(4aS,7aR)-1-(3-hydroxypyridine-2-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2-ethoxypyridin-3-yl)methyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
5-({2-[2-(1-phenylethyl)-1H-imidazol-1-yl]ethyl}sulfanyl)-1H-1,2,3-triazole
(4aR,8aR)-2-methanesulfonyl-7-{[4-(methylsulfanyl)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
2-methyl-5-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
(1S,9aR)-1-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-octahydro-1H-quinolizine
4-{1-[(2,5-dimethoxyphenyl)methyl]piperidin-4-yl}-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
6-methyl-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-[6-hydroxy-4-(5-methyl-1,2-oxazole-3-carbonyl)-1,4-diazepan-1-yl]pyridine-3-carbonitrile
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2-(methylamino)ethan-1-one
2-(2-methoxyphenoxy)-N-[(1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}piperidin-3-yl)methyl]acetamide
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
2-(5-acetylthiophen-3-yl)-N-[(2,3,4-trifluorophenyl)methyl]acetamide
3-[1-(furan-2-ylmethyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
2-[(3aS,6aS)-3a-(methoxycarbonyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]acetic acid
1-(3-ethoxybenzoyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
(1R,9S)-5-amino-3-[4-hydroxy-3-methoxy-5-(prop-2-en-1-yl)phenyl]-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]acetamide
1-(3-chlorobenzoyl)-4-propyl-1,4-diazepan-5-one
3-(1-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(3-fluorophenyl)urea
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]urea
(1R,9aR)-1-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-ylmethyl}-octahydro-1H-quinolizin-1-ol
2-(3-methoxypropyl)-1-[4-(pyrrolidin-1-ylmethyl)benzoyl]piperidine
2-{[(1-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
4-ethyl-1-[(4-methanesulfonylphenyl)methyl]-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonitrile
3-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidine-1-carbonyl]-8-methyl-1,4-dihydroquinolin-4-one
2-[4-(pyrrolidine-1-carbonyl)phenyl]pyridine-3-carbonitrile