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1-cyclopropyl-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-5-oxopyrrolidine-3-carboxamide
3-{3-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]propyl}-1H-indole
6-[4-(1-ethoxyethyl)phenyl]-N,N-dimethylpyridazin-3-amine
1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
1-(2-methoxy-5-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
3-(methanesulfonylmethyl)-5-{[4-(propan-2-yl)phenyl]methyl}-1,2,4-oxadiazole
2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1-(morpholin-4-yl)ethan-1-one
methyl (2S,4R)-1-methyl-4-(2,3,4,9-tetrahydro-1H-carbazole-7-amido)pyrrolidine-2-carboxylate
(2S)-2-{[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]formamido}-4-methylpentanoic acid
(2S)-2-amino-N-[2-(dimethylamino)ethyl]-3-phenyl-N-(thiophen-3-ylmethyl)propanamide
2-[(4-methylpiperidin-1-yl)methyl]-4-(pyrimidin-2-yl)phenol
5-methyl-1-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-benzyl-3-ethyl-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-1,4-diazepan-5-one
1-(5-{[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
3,3-dimethyl-1-{2-[3-(2-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}urea
2-(2-{[2-(5-methylfuran-2-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1'-(3,6-dimethyl-1-benzofuran-2-carbonyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(3-{2-[2-(ethylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}phenyl)acetamide
2-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidine-1-carbonyl]benzonitrile
N-butyl-2-(propan-2-yloxy)-N-(thiophen-3-ylmethyl)propanamide
4-[2-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]-5-methyl-2,3-dihydro-1H-pyrazol-3-one
N-cyclopropyl-4-methoxy-3-{[1-(1,3-oxazole-5-carbonyl)piperidin-4-yl]oxy}benzamide
2,6-dimethoxy-4-[(4-{2-[(2-methylphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)methyl]phenol
N-(3-cyano-4-methylphenyl)-4-hydroxy-4-phenylpiperidine-1-carboxamide
7-cyclohexyl-2-(5-ethyl-1H-pyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
6-[(4-ethylphenyl)methyl]-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
N-ethyl-7-[(4-fluorophenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
8-chloro-2-(furan-2-yl)-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]quinoline-4-carboxamide
2-[5-(1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
(3S,7S)-5-(2-oxo-2-phenylacetyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
4-{[5-(oxan-2-yl)furan-2-yl]methyl}piperazine-1-sulfonamide
N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-2-methylimidazo[1,2-a]pyridine-6-carboxamide
2-(2-aminoethyl)-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]quinazolin-4-amine
2-(2-methoxyethyl)-8-[3-(4-methylpiperazin-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
(3S)-1-ethyl-4-(3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanoyl)-3-methylpiperazin-2-one
1-[9-(but-3-yn-1-yloxy)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
4-{[2-(1H-indol-3-yl)ethyl]amino}-5-methyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(2-phenoxyethyl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
2-[(dimethylcarbamoyl)amino]-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1-benzothiophene-2-carboxamide
8-[(2E)-3-(5-chloro-2-hydroxyphenyl)-2-methylprop-2-en-1-yl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}isoquinoline-1-carboxamide
2-methoxy-5-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}pyridine
4-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-6-methylpyrimidin-2-amine
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-[(6-methylquinolin-5-yl)methyl]acetamide
2,3-dimethyl-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)quinoxaline-6-carboxamide
N-[2-(3-chlorophenyl)ethyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
6-(2-methylpropyl)-2-oxo-N-[3-(pyridin-3-yl)propyl]-1,2-dihydropyrimidine-4-carboxamide
1-{4-[(2S)-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one