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N-[(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-3-phenyl-1H-pyrazole-5-carboxamide
(3S,4S)-1-(4-amino-5-methylpyrimidin-2-yl)-4-(2H-1,3-benzodioxol-5-yl)piperidin-3-ol
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-{[3-(methylsulfanyl)phenyl]methyl}piperidine
3-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-ylmethyl}-4,5,6,7-tetrahydro-1,2-benzoxazole
(1R,3S)-7-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-7-azaspiro[3.5]nonane-1,3-diol
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]pyridin-2-amine
3-[(dimethylamino)methyl]-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-3-ol
methyl 2-[1-(benzylsulfamoyl)-3-oxopiperazin-2-yl]acetate
7-methoxy-3-{[3-(morpholin-4-yl)phenyl]methyl}-2,3,4,5-tetrahydro-1H-3-benzazepine
2-{4-[1-(dimethylamino)ethyl]phenyl}-6-methylpyridine-3-carboxamide
4-[(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)methyl]-N-methylbenzene-1-sulfonamide
4-[(2S)-2-(3-ethyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]pyridine
4-ethyl-3-{1-[2-(1H-indol-1-yl)acetyl]piperidin-3-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-ethyl-2-{4-[4-(propan-2-yl)benzoyl]piperazin-1-yl}acetamide
1-[3-(1H-imidazol-1-yl)propyl]-2-(1-methyl-1H-imidazol-2-yl)-1H-imidazole
3-(furan-2-ylmethyl)-3-(1-hydroxybutan-2-yl)-1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]ethan-1-one
1-(benzenesulfonyl)-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperazine
2-[(1-benzyl-1H-imidazol-5-yl)methyl]-2-azaspiro[4.5]decan-3-one
N-[3-(4-methoxyphenyl)propyl]-6-(pyridin-4-yl)pyridine-3-carboxamide
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(3-methylthiophen-2-yl)methyl]amine
N-(3-hydroxypropyl)-1-(1-{[3-(2-methylphenyl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
4-[2-(3-chlorophenyl)-2-hydroxyacetyl]-1-(4-methylphenyl)piperazin-2-one
naphthalen-1-yl (7S,9aR)-6,9-dioxo-7-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-3-azaspiro[5.5]undecan-9-amine
N-(3-chloro-4-methoxyphenyl)-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
2-(dimethylamino)-N-methyl-N-{2-phenyl-1-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]ethyl}acetamide
3-(dimethyl-1H-1,2,4-triazol-1-yl)-N,2-dimethyl-N-[(3-methylthiophen-2-yl)methyl]propanamide
1-[(5-methylfuran-2-yl)methyl]-4-oxo-5-(4-phenylazepane-1-carbonyl)-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
{1-[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}(pyridin-3-yl)methanol
N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]propan-1-one
5-chloro-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
1-[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]-2-(oxan-2-ylmethoxy)ethan-1-one
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-[(3-fluorophenyl)methyl]acetamide
N-[2-methyl-1-(pyridin-3-yl)propyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-(2-hydroxyethyl)-9-[(3-phenyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-methanesulfonyl-2-{[3-(5-methylfuran-2-yl)-1H-pyrazol-5-yl]formamido}butanoic acid
(3S,4R)-N,N-dimethyl-1-(1-methyl-1H-indazole-3-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-amine
2-{4-[3-(4-fluorophenoxy)propyl]piperazine-1-carbonyl}-1-methylazepane
2-(adamantan-1-yl)-4-hydroxy-N-[(5-methyl-1,2-oxazol-3-yl)methyl]pyrimidine-5-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
7-fluoro-3-[2-(piperazin-1-yl)ethyl]-3,4-dihydroquinazolin-4-one
2-(3-methyl-1,2-oxazol-5-yl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-(5-{[5-(2-chlorophenyl)furan-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
1-(5-methoxyfuran-2-carbonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(3R,5S)-N-[3-(dimethylamino)propyl]-1-(2-methylpropyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
1-{2-methylthieno[3,2-d]pyrimidin-4-yl}-4-(4H-1,2,4-triazol-4-yl)piperidine