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(3R,4R)-1-(5-methoxy-2,4-dimethylbenzenesulfonyl)-3,4-dimethylpyrrolidin-3-ol
3-(3-hydroxy-1,2-oxazol-5-yl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)propanamide
{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-2-phenylethyl}[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
2,2,6,6-tetramethyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]piperidin-4-amine
3-hydroxy-3-{[4-(2-hydroxyethyl)piperidin-1-yl]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-(5-fluoroquinolin-8-yl)-N,N-dimethylpyrimidin-4-amine
2-(3-fluoro-2,4-dimethylphenyl)-1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazole
{4-[(4-chlorophenyl)methyl]-1-[4-(propan-2-yloxy)benzoyl]piperidin-4-yl}methanol
1-[1-(pyrazin-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
7-(7-fluoro-4-methylquinolin-2-yl)-4-(2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,N-dimethyl-2-{9-oxo-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-2-yl}acetamide
3-[(3R,4S)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-[3-benzyl-3-(hydroxymethyl)piperidin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
2-[(2E)-3-phenylprop-2-en-1-yl]-8-(propane-1-sulfonyl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-(1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-4-yl)ethyl]acetamide
N-(4-methylphenyl)-N-(2-{2-oxa-7-azaspiro[4.5]decan-7-yl}-2-oxoethyl)methanesulfonamide
({5-benzoyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)(methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-[7-(3-methoxypropyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-4,6-dimethylpyridine-3-carbonitrile
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]pyrrolidin-3-yl]methanol
2-acetyl-8-(3-methoxypyrazin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[4-(1,4-dithiepan-6-yl)-1-[(2-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(4,4,4-trifluorobutyl)-2,8-diazaspiro[4.5]decan-3-one
1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3-[3-(propan-2-yloxy)benzoyl]piperidine
1-(3-{3-[(3-methylphenyl)methyl]-1,2,4-oxadiazol-5-yl}propyl)piperidine
1-[2-methyl-3-(pyrrolidin-1-yl)phenyl]-3-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}urea
8-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
1-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-indole-2-carboxamide
N-[(3S,4R)-1-(2-methoxyquinoline-4-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
1-[(2-ethylphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-cyclopropyl-6-(1,2,3,4-tetrahydronaphthalen-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}(pyridin-2-yl)methanol
2-{4-[(4-methylphenyl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
1-(cyclohexylmethyl)-5-(diethylamino)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
8-(2-hydroxy-4-methylpentanoyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[3-(methylsulfanyl)propyl]-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
3,5-dimethoxy-2-{[(2S)-4-methyl-2-(propan-2-yl)piperazin-1-yl]methyl}benzoic acid
2-{4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
5-(azepane-1-carbonyl)-1-(butan-2-yl)-4-oxo-N-{[2-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
N-[3-(1,3-benzothiazol-2-yl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
9-(4-fluoro-3-methylbenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{1-butyl-5-[2-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazol-3-yl}pyridine
1,7-dimethyl-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-indole-2-carboxamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}-N-ethylcyclopropanamine
3-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)-1-(4-phenylpiperazin-1-yl)propan-1-one
N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-N-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
(3S,4R)-N,N-dimethyl-1-[3-(piperidine-1-carbonyl)pyridin-2-yl]-4-propylpyrrolidin-3-amine