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2-methyl-6-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-ethyl-4-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-[2-(furan-2-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{3-[({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}amino)methyl]phenoxy}-3-(morpholin-4-yl)propan-2-ol
2-methyl-1-[3-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]propan-1-one
(3aR,5R,6S,7aS)-2-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}-octahydro-1H-isoindole-5,6-diol
7-(2-methoxyethyl)-2-(2-methylpyridin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-methoxypropyl)acetamide
1-(2-{[2-(azepan-1-yl)ethyl](methyl)amino}pyrimidin-4-yl)pyrrolidin-3-ol
1-{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-4-yl}piperidin-4-ol
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-methyl-2-[(2S)-2-(methylamino)propanoyl]-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-({ethyl[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)-4-methylphenol
3-(2-ethoxyethyl)-1-methyl-5-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-1,2,4-triazole
5-{[2-(2-cyclohexyl-1H-imidazol-1-yl)ethyl]sulfanyl}-1H-1,2,3-triazole
N-[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-amine
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[3-(1H-pyrazol-1-yl)phenyl]methyl})amine
5-(3,4-dimethylphenoxymethyl)-N-(1H-indol-2-ylmethyl)-1,2-oxazole-3-carboxamide
1-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyphenyl)piperazine
2-(1-{[3-(5-methylfuran-2-yl)phenyl]methyl}azetidin-3-yl)pyridine
5-cyano-2-methyl-6-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyridine-3-carboxylic acid
3-[({1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}oxy)methyl]pyridine
N-[1-(1-acetylpiperidin-4-yl)-1H-pyrazol-5-yl]-2H-1,3-benzodioxole-5-carboxamide
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-(3-phenyl-1H-pyrazol-1-yl)acetamide
dimethyl({[(3R,4S)-4-propyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl]sulfamoyl})amine
N-(1-{1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
N-(1H-imidazol-2-ylmethyl)-2-[4-methyl-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]acetamide
N-(oxolan-3-ylmethyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
(3R)-3-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1-({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)-3-methylpiperidin-3-ol
methyl 2-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxylate
[3-(2,5-dimethylphenoxy)propyl](methyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
1-(cyclohexyloxy)-3-[5-(furan-3-yl)-4-phenyl-1H-imidazol-1-yl]propan-2-ol
[(1-cyclohexylpiperidin-3-yl)methyl][(4-fluoro-3-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
N-[(5-chlorothiophen-2-yl)methyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
methyl (2S)-2-{[5-(4-methylpiperidine-1-carbonyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridin-3-yl]formamido}-2-phenylacetate
4-(furan-3-yl)-5-[(4-methoxy-2,3-dimethylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
7-(2-cyclohexylethyl)-2-(1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(3-methoxyphenyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)acetamide
3-(1,3-benzothiazol-2-yl)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}propan-1-one
(2R)-3-methyl-2-({4-[(6-methylpyridin-3-yl)oxy]piperidin-4-yl}formamido)butanamide
5-(dimethylamino)-2-{[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dihydropyridazin-3-one
(3S,4S)-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-4-(naphthalen-2-yl)piperidin-3-ol
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(3-fluorophenyl)methyl]urea
N-(2-{7-[(2,6-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-fluorobenzamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-2-(ethylamino)pyrimidine-5-carboxamide
2-methyl-N-(2-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridin-3-yl)propanamide