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N-(1H-1,3-benzodiazol-2-yl)-2-{3-[3-(1-methyl-1H-imidazol-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
1-[3-(thiomorpholine-4-carbonyl)phenyl]imidazolidin-2-one
3-methoxy-2-[4-(2-methoxyethoxy)phenyl]pyridin-4-amine
N,1-dimethyl-2-oxo-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}imidazolidine-4-carboxamide
2-phenoxy-1-{4-[4-(pyridin-3-yl)pyrimidin-2-yl]piperazin-1-yl}ethan-1-one
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(propan-2-yloxy)ethan-1-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]acetamide
3-(3-hydroxy-3-methylbutyl)-N-(1,3-thiazol-2-ylmethyl)benzamide
1-[2-(dimethylamino)ethyl]-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
5-{[2-(benzyloxy)phenyl]methyl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-[1-(2-aminopyrimidin-4-yl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
6-fluoro-2-methyl-N-[2-(piperidin-1-yl)ethyl]quinoline-4-carboxamide
(2R)-2-({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)propanamide
3,5-dimethoxy-N-{1,8,15-triazatetracyclo[7.6.0.03,7.010,14]pentadeca-2,7,9,14-tetraen-2-yl}benzamide
methyl 1-(2-hydroxy-3-{3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}propyl)piperidine-4-carboxylate
2-({1-methyl-9-pentanoyl-1,4,9-triazaspiro[5.5]undecan-4-yl}methyl)benzonitrile
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
1-(3,4-dimethoxyphenyl)-3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]urea
3-(4-tert-butylbenzoyl)-1-(oxan-4-yl)piperidine
2-[(2-chlorophenyl)methyl]-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyridin-2-amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
2-[2-(butan-2-yloxy)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-(pyridin-3-ylmethyl)propanamide
5-(methoxymethyl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)furan-2-carboxamide
4-(hydroxymethyl)-1-(1,3-thiazol-2-ylmethyl)azepan-4-ol
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[1-(pyridin-3-yl)propan-2-yl]acetamide
1-(thiophen-2-ylmethyl)-5-(2,4,5-trimethoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-(3-fluorophenyl)-N-[(3-methyl-1-phenyl-1H-1,2,4-triazol-5-yl)methyl]methanesulfonamide
3-[5-(2,6-dimethoxyphenyl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
(3aS,6aR)-N-(furan-2-ylmethyl)-3-[(2-methoxyphenyl)methyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-methyl-1H-pyrazole-5-carboxamide
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[2-(pyridin-2-yl)ethyl]amine
3-benzyl-1-methyl-3-[2-oxo-2-(1,2,3,6-tetrahydropyridin-1-yl)ethyl]-2,3-dihydro-1H-indol-2-one
N-[(2S,4R,6R)-2-(3-chloro-4-hydroxyphenyl)-6-cyclohexyloxan-4-yl]acetamide
7-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
3-(6-methoxynaphthalene-2-carbonyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
1-(3-ethoxy-2-hydroxypropyl)-5,5-diphenylpiperidin-2-one
4-(2-methylphenoxy)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidine-4-carboxylic acid
4-[3-(2-methoxyethyl)-5-(morpholin-2-yl)-1H-1,2,4-triazol-1-yl]-1-methyl-1,2-dihydroquinolin-2-one
3-[3-(2-methoxyethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-2-(methylsulfanyl)pyridine
2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
3-(2,5-dioxoimidazolidin-4-yl)-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
5-(3,4-dimethylphenoxymethyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
1-[(3-fluoro-4-hydroxy-5-methoxyphenyl)methyl]-4-(2-methylquinolin-6-yl)piperidin-4-ol
4-{4-[3-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]piperidine-1-carbonyl}imidazolidin-2-one
1-(2-{8-chloro-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl}ethyl)-1H-pyrazole
4-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
5-({3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)-1,3-oxazolidin-2-one
(3aR,6aR)-2-cyclopentyl-N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide