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4-{3-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
[(6-fluoroquinolin-2-yl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
1-(3-methoxybenzoyl)-4-[(2S)-pyrrolidine-2-carbonyl]piperazine
2-[(4aS,8aR)-2-oxo-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-6-yl]pyridine-3-carbonitrile
1-{4-[2-(cyclohexylmethyl)morpholine-4-carbonyl]piperidin-1-yl}ethan-1-one
2-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-6-fluoro-1H-1,3-benzodiazole
3-(2,5-dioxoimidazolidin-4-yl)-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]propanamide
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-5-ethyl-1,3-oxazole-4-carboxamide
1-cyclopentanecarbonyl-4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-({3-cyclopropyl-1-[2-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}methyl)-1H-1,2,3,4-tetrazole
1-[benzyl(methyl)amino]-3-[4-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
3-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-1,4-dihydropyridin-4-one
1-(2,3-dihydro-1H-inden-2-yl)-N-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-(2-oxo-1,2-dihydropyridin-1-yl)propanamide
(4aR,7aS)-1-(2-hydroxyethyl)-4-[2-(4-hydroxyphenyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(3-chlorophenyl)-8-oxo-N-(oxolan-3-ylmethyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-[(2-methylphenyl)sulfanyl]acetamide
7-[(2,3-dimethoxyphenyl)methyl]-6-oxo-N-(prop-2-en-1-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
3-chloro-6-[2-ethoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridazine
N-[(2-methylphenyl)methyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
8-(2-methylbenzoyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1S,5R)-3-[2-(benzyloxy)ethyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
N-methyl-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(1-phenylpyrrolidin-3-yl)methyl]acetamide
2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrazine
(2S,3R)-2-{[2-(2,3-difluorophenoxymethyl)-1,3-oxazol-4-yl]formamido}-3-hydroxybutanamide
[(3-ethoxyphenyl)methyl]({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
3-{1-[2-(4-methoxyphenyl)acetyl]piperidin-4-yl}-N-phenylpropanamide
N1,N1-dimethyl-N4-[(5-methylpyrazin-2-yl)methyl]piperidine-1,4-dicarboxamide
3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-methyl-2-[(2-methylphenyl)methyl]-1-(pyridin-4-ylmethyl)-1,4-dihydropyridin-4-one
[(3S,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(2-methylpyrimidin-4-yl)piperidin-3-yl]methanol
(2S,4R)-4-amino-N-methyl-1-[(4-methylphenyl)methanesulfonyl]pyrrolidine-2-carboxamide
1-methyl-3-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]-1H-indazole
N-(1-{4-[(1,4-dioxan-2-ylmethyl)carbamoyl]phenyl}-1H-pyrazol-4-yl)-2,4-dimethylbenzamide
2-methyl-9-[2-(2-methyl-1H-imidazol-1-yl)acetyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[2-(propan-2-ylsulfanyl)ethyl]piperidine
{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}({[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl})amine
3-(3,4-dimethoxybenzoyl)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidine
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(6-methylpyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,3R)-3-[3-(1H-1,2,3,4-tetrazol-1-yl)propanamido]-N-[2-(thiophen-2-yl)ethyl]cyclopentane-1-carboxamide
4-methyl-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1,4-diazepan-5-one
2-(1,2-benzoxazol-3-yl)-N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]acetamide
2-amino-1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
3-(2,5-dioxoimidazolidin-4-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]propanamide
1-methyl-4-({5-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
7-(cyclobutylmethyl)-2-[3-(thiophen-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
8-methyl-N-[(3-methylphenyl)methyl]-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
2-[1-(2,3-dihydro-1-benzofuran-7-carbonyl)-1,4-diazepan-6-yl]acetic acid