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ethyl 1-(prop-2-en-1-yl)-5-(1,3-thiazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-acetamido-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}propanamide
methyl 9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-3-{[4-(methylsulfanyl)phenyl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(2-fluorophenyl)-N-{2-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}acetamide
N-[(4-methanesulfonylphenyl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
N-[2-(4-methylphenyl)ethyl]-3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
N-{[1-(1,4-dithiepan-6-yl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide
1-[2-(methylamino)pyridine-4-carbonyl]-N-[4-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(1S,4S)-2-(2-fluorophenyl)-5-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
(1S,4R)-4,7,7-trimethyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-3-oxo-2-oxabicyclo[2.2.1]heptane-1-carboxamide
4-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)morpholine
1-[(3-fluorophenyl)methyl]-6-oxo-N-{2-[4-(propan-2-yloxy)phenyl]ethyl}piperidine-3-carboxamide
N-(1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)acetamide
{[(3S,4R)-1-(5-fluoropyridine-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-(furan-2-ylmethyl)-3-methoxy-N-(3-methylbutan-2-yl)propanamide
1-(diethylamino)-3-[2-methoxy-4-({[2-(6-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-(4-{[3-(hydroxymethyl)-3-propylpiperidin-1-yl]methyl}phenoxy)-1-(pyrrolidin-1-yl)ethan-1-one
5-(2-chlorophenyl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]furan-2-carboxamide
3-({[2-(2-amino-1,3-thiazol-4-yl)ethyl]amino}methyl)piperidin-3-ol
9-[(5-ethylpyridin-2-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
(4-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenyl)methanol
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-1H-pyrazole-3-carboxamide
1-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(propan-2-yloxy)ethan-1-one
3-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]phenol
3-cyclohexyl-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}propan-1-one
3-{2-[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,3-oxazinan-2-one
1-(1-{5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidin-4-yl)piperidin-4-ol
2-(2,3-dihydro-1H-inden-5-yloxy)-N-[(4-hydroxyazepan-4-yl)methyl]-2-methylpropanamide
1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]piperidin-4-amine
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-[(4-methylpiperidin-1-yl)sulfonyl]pyrrolidin-3-amine
1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-{1-oxaspiro[4.4]nonan-3-yl}urea
2-chloro-N-(2-{[(2R,4R)-4-hydroxypyrrolidin-2-yl]formamido}ethyl)benzamide
1-(2,6-difluoro-3-methylbenzoyl)-2-(pyrrolidine-1-carbonyl)piperazine
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-3-{[4-(methylsulfanyl)phenyl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-4-methyl-2-(propan-2-yl)-1,3-thiazole
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(1H-pyrazol-1-yl)propan-1-one
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
7-fluoro-3-methyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1-benzofuran-2-carboxamide
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-[1-(thiophen-2-yl)propan-2-yl]benzamide
3-hydroxy-S-[2-(2-hydroxybenzoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]butane-1-sulfonamido
1-phenyl-5-[5-(pyrrolidin-1-ylmethyl)furan-2-yl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
4-ethyl-1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-4-methylpiperidine
4-ethyl-3-{1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N,N-diethyl-2-{4-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}acetamide
(3S,5R)-1-(3,3-dimethylbutanoyl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid