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4-[(4-cyclopentylpyrimidin-2-yl)amino]-1-[(3-fluorophenyl)methyl]pyrrolidin-2-one
N-(1-benzylpiperidin-4-yl)-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-methoxy-5-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
2-[5-(dimethoxy-1,3,5-triazin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1H-1,3-benzodiazole
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
5-chloro-N-[(3R,4S)-1-cyclopentyl-4-cyclopropylpyrrolidin-3-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
N,N,2-trimethyl-7-(3-phenyl-1H-pyrazole-4-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
6-{[(3S)-3-ethylmorpholin-4-yl]sulfonyl}-1,2,3,4-tetrahydroquinoxaline-2,3-dione
5-ethyl-N,2-dimethyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]pyrimidin-4-amine
(1R,5R)-3-cyclobutanecarbonyl-6-[(3,5-dichloropyridin-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(3,3-diphenylpiperidin-1-yl)-3-(morpholin-4-yl)propan-1-one
2-methyl-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1,3-thiazole-5-carboxamide
6-(dimethylamino)-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]pyridine-3-carboxamide
6-(3-fluorophenyl)-N-methyl-N-(1-methylpyrrolidin-3-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(3S)-4-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-3-ethylmorpholine
2-amino-4-[4-(3-hydroxyprop-1-yn-1-yl)phenyl]-6-(4-methyl-1,3-thiazol-5-yl)pyridine-3-carbonitrile
5-benzyl-1-(4-methylphenyl)-4-(1H-pyrazole-3-carbonyl)piperazin-2-one
6-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)-1H-imidazol-1-yl]-3-methyl-2,3-dihydro-1,3-benzoxazol-2-one
7-(cyclobutylmethyl)-2-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2,7-diazaspiro[4.5]decan-6-one
1-(azepan-1-yl)-3-(2-methoxy-4-{[(oxan-4-yl)amino]methyl}phenoxy)propan-2-ol
N-{4-[4-(4-cyclopentylpiperazin-1-yl)piperidin-1-yl]phenyl}-2-(3-fluorophenyl)acetamide
2,3-dimethyl-6-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}quinoxaline
1-cyclopentyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-6-oxopiperidine-3-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-5-chlorothiophene-2-carboxamide
2-(4-phenylpiperidin-1-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]ethan-1-one
2-(3-methoxyphenyl)-1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-methyl-4-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-5-propylpyrimidine
3-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-3,4-dihydroquinazoline-7-carboxamide
(3R,5S)-N-[3-(dimethylamino)propyl]-1-(2-methylpropyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}piperidine-3-carboxamide
N-({5-fluoro-7-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-4-(thiophen-2-yl)butanamide
1-[(2E)-3-phenylprop-2-en-1-yl]-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazine
N-ethyl-3-(4-hydroxyphenyl)-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
2-{[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](ethyl)amino}-N-(1,3-thiazol-2-yl)propanamide
5-propyl-4-{4-[4-(pyrazin-2-yl)piperazin-1-yl]piperidin-1-yl}pyrimidine
5-(methoxymethyl)-N-(3-methyl-1-{7-[(3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)furan-2-carboxamide
8-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-chloro-3-[3-(2-hydroxypropan-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-6-methylpyridine-3-carbonitrile
2-(cyclohexylmethyl)-4-[4-(1H-pyrazol-3-yl)benzoyl]morpholine
4-(hydroxymethyl)-1-(6-methyl-2-propylpyrimidin-4-yl)azepan-4-ol
2-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-ol
1-[5-(2-methylphenyl)-1,2,4-triazin-3-yl]-4-phenyl-1,4-diazepane
N-ethyl-3-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-cyclopentyl-1,4-diazepane
3-(2-oxopiperidin-1-yl)-N-[(1R)-2,2,2-trifluoro-1-phenylethyl]propanamide
4-[2-(1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-2-yl)ethyl]phenol
(2S)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-N-ethylpyrrolidine-2-carboxamide
5-[(3,5-dichloropyridin-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,2-dimethyloxan-4-amine