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N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-7-fluoro-2-methylquinoline-4-carboxamide
(3S)-3-methyl-1-(2-methylpropyl)-4-{4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanoyl}piperazin-2-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-N-(6-chloropyridin-3-yl)-3-hydroxypiperidine-1-carboxamide
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-[(4-methylphenyl)sulfanyl]propanamide
N4-cyclopropyl-N6-(pyridin-2-ylmethyl)pyrimidine-2,4,6-triamine
3-methyl-7-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
methyl 2-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)piperidine-1-carboxylate
(3S,4S)-1-(2-{[(4-chlorophenyl)methyl]carbamoyl}ethyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-[2-(2-methoxyphenyl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-(propan-2-yl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-1H-pyrazole-4-carboxamide
N-[(2-ethoxypyridin-3-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-propyl-1H-pyrazol-3-yl)methyl]amine
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(pyridazine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3S,4S)-4-cyclopropyl-1-({1-methyl-4-oxo-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-6-yl}methyl)pyrrolidine-3-carboxylic acid
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetamide
5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
2-{1-[3-(1H-imidazol-2-yl)benzoyl]azetidin-3-yl}pyridine
2-(1-methyl-1H-pyrrol-3-yl)-1-{4-[4-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
5-{4-hydroxy-1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
N-[(2-aminopyridin-3-yl)methyl]-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-({3-methanesulfonylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-N-methyl-1,2,3,4-tetrahydronaphthalen-1-amine
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]methylamine
8-(5-chloropyridine-2-carbonyl)-2-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[(4-methoxyphenyl)methyl]-4-[2-(morpholin-4-yl)propanoyl]piperazin-2-one
6-methyl-5-[5-(1-methyl-1H-pyrazol-5-yl)-1,2,4-oxadiazol-3-yl]-2-(1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
2-[4-(hydroxymethyl)phenyl]-2-[methyl(oxan-4-ylmethyl)amino]acetic acid
4-benzyl-3-ethyl-1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-1,4-diazepan-5-one
dimethyl({2-[1-(5-phenyl-1,3-oxazole-4-carbonyl)piperidin-2-yl]ethyl})amine
N-ethyl-9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
N-cyclopentyl-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-amine
5-[3-(4-phenylpiperazin-1-yl)piperidine-1-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
4-(1-{1-[1-(2-fluorophenyl)propan-2-yl]piperidin-4-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
N-[1-({[3-(1H-indol-1-yl)propyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
2-(4-fluoro-3-methylphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-2-(pyrimidin-2-ylsulfanyl)acetamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)pyrrolidin-3-yl]methanol
N-(3-chloro-4-methoxyphenyl)-4-(oxan-4-yl)piperazine-1-carboxamide
ethyl 1-[(5-chloro-2-hydroxyphenyl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylate
3-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
2-cyclopropyl-8-[4-(4-methylphenyl)-4-oxobutyl]-2,8-diazaspiro[5.5]undecan-3-one
2-{[(2-amino-1,3-thiazol-4-yl)methyl]amino}-N-[(4-acetamidophenyl)methyl]acetamide
3-{2-oxo-2-[2-(3-phenylpropyl)morpholin-4-yl]ethyl}-1,2,3-oxadiazol-3-ium-5-olate
3,3-diphenyl-1-(1H-1,2,4-triazole-5-carbonyl)piperidine
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
methyl 3-[(3,5-difluorophenyl)methyl]-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)quinoline-8-sulfonamide
4-[1-(pyridin-3-yl)-2-(4H-1,2,4-triazol-4-yl)ethyl]morpholine
1-(cyclopropylmethyl)-4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2-(propan-2-yl)-1,4-diazepane
2-methoxy-1-(4-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one