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(2-{[4-(1-methyl-1H-indole-2-carbonyl)piperazin-1-yl]methyl}phenyl)methanol
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
3-methyl-3-[3-(oxolan-2-yl)propyl]-1-{3-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}urea
4-(1H-indazol-5-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(2,1,3-benzothiadiazol-5-ylmethyl)({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl})(2-methoxyethyl)amine
N-{1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-hydroxy-1-oxopropan-2-yl}acetamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-1H-pyrrole-3-carboxamide
3-(piperidine-1-carbonyl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]benzene-1-sulfonamide
ethyl 3-(2-methoxyethyl)-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine-3-carboxylate
1-(3-methoxypropyl)-4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(5-methylfuran-2-yl)ethyl]benzamide
3-(3-hydroxy-3-methylbutyl)-N-[(3-hydroxyphenyl)methyl]-N-methylbenzamide
methyl({[3-(2-methylphenyl)phenyl]methyl}){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
6-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-(3-benzoylpiperidine-1-carbonyl)thiophene-3-sulfonamide
1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-4-(oxolan-2-ylmethyl)piperazine
2-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-2-yl)acetamide
2-(azepan-1-yl)-1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]ethan-1-one
N-(2-hydroxyethyl)-5-{1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-ethyl-4-[(pentan-3-yl)amino]pyrrolidin-2-one
(4aS,8aR)-1-(carboxymethyl)-6-[(3-fluorophenyl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
(1R,7S)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(3-methylbutyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
6-tert-butyl-1-methyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[({2-methylthieno[3,2-d]pyrimidin-4-yl}amino)methyl]-1H-1,2,4-triazol-5-amine
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
1-(3,5-difluorophenyl)-N-{[3-(methylsulfanyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-(1H-imidazol-1-yl)-1-[6-(piperidin-1-yl)pyrimidin-4-yl]piperidine-4-carboxylic acid
9-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(adamantane-1-carbonyl)-4-[2-(pyrrolidin-1-yl)ethyl]-1,4-diazepan-5-one
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
4-[3-(3-fluorophenyl)-1H-pyrazol-4-yl]-3-methyl-4H,5H,6H,7H-[1,2]thiazolo[5,4-b]pyridin-6-one
3-[(2,1,3-benzothiadiazol-5-ylmethyl)(ethyl)amino]-1λ6-thiolane-1,1-dione
2-cyclopentyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}acetamide
N-cyclopropyl-4-{[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]sulfamoyl}benzamide
9-[4-(4-methylpyridin-2-yl)piperazin-1-yl]-3-azaspiro[5.5]undecane
13-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
5-({[2-(dimethylamino)ethyl][(2-methylphenyl)methyl]amino}methyl)-2-methoxyphenol
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-(4-fluorobutyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-N-[(3-methylthiophen-2-yl)methyl]cyclopentanamine
4-chloro-N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
(1R,5R)-6-(cyclobutylmethyl)-3-(3-methyl-1,2-oxazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
(3S,4S)-1-{imidazo[1,2-a]pyridine-6-carbonyl}-4-methylpiperidine-3,4-diol
1-(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
(1R,7S)-3-(3,4-dimethylphenyl)-N-methyl-4-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-methyl-6-[5-(oxolan-3-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]-1,3-benzothiazole
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
5-(4-cyclobutanecarbonyl-1,4-diazepane-1-carbonyl)-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one