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N-[(4-chlorophenyl)methyl]-3-[(3S,4R)-3-acetamido-4-propylpyrrolidin-1-yl]propanamide
1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-[2-(thiophen-2-yl)ethyl]piperidine
3-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propanamide
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-{[4-(5-methylfuran-2-yl)phenyl]methyl}piperidin-4-ol
N-(2-{7-[(4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N,3-dimethyl-4,5-dihydro-1,2-oxazole-5-carboxamide
3-[3-(4-methylpiperazin-1-yl)propyl]-1-[3-(1H-pyrazol-5-yl)phenyl]urea
N-[2-(3-hydroxypiperidin-1-yl)ethyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
3-(oxolan-3-yl)-5-[3-(1H-pyrazol-4-yl)propyl]-1,2,4-oxadiazole
1-(2-methoxyethyl)-N-[2-(2-methylphenyl)ethyl]-6-oxopiperidine-3-carboxamide
3-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[(4-ethylphenyl)methyl]methylamine
N-[(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}pyrrolidin-3-yl)methyl]methanesulfonamide
{[(3S,4R)-1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-[3-(1H-pyrazol-1-yl)azetidin-1-yl]pyridine-3-carboxamide
5-(methoxymethyl)-N-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
1-({5-[1-(ethanesulfonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)azepane
1-methyl-N-(2-phenylethyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
9-[3-(4-hydroxyphenyl)propanoyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-1-[(3-methoxyphenyl)methyl]-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-3-{methyl[(1-methyl-1H-indol-2-yl)methyl]amino}butanamide
5,6-dimethyl-2-oxo-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
2-methyl-3-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1,2,3,4-tetrahydroisoquinoline
3-(2-chloro-5-sulfamoylphenyl)-1-(oxan-4-yl)urea
4-methyl-2-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenol
5-(propan-2-yl)-N-{3-[(pyridin-3-yl)amino]propyl}-1,2-oxazole-3-carboxamide
4-[(4aS,7aR)-4-(3-methylbutanoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]benzonitrile
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(4-methanesulfonylmorpholin-2-yl)methyl]acetamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
(3R,4S)-4-(4-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-diazepan-1-yl)oxolan-3-ol
methyl 1-({3-[(1-methyl-1H-imidazol-2-yl)carbamoyl]phenyl}methyl)piperidine-4-carboxylate
4-ethyl-3-{1-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-oxoethyl]-1,2-dihydropyrimidin-2-one
1-{1-[(2,6-difluorophenyl)methyl]piperidin-3-yl}-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
1-ethyl-N-[2-(2-phenoxyethoxy)phenyl]-1H-pyrazole-4-carboxamide
1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-propoxypiperidine
1-[(2S)-oxolane-2-carbonyl]-4-[4-(piperidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-5-(3-methyl-1,2-oxazol-5-yl)furan-2-sulfonamide
1-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
1-benzyl-3-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
4-{3-[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]propoxy}benzamide
4-ethyl-1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-chloro-5-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-[2-(4-chlorophenyl)-2-(piperidin-1-yl)ethyl]-4-hydroxy-2-methylpyrimidine-5-carboxamide
{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}({[1-(pyrimidin-2-yl)piperidin-3-yl]methyl})amine
(cyclopropylmethyl)({[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
6-[(diethylamino)methyl]-N-[3-(propan-2-yl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
9-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
4-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1H-imidazol-2-yl}-5-methyl-2-(thiophen-2-yl)-1,3-oxazole