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2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
[(1-ethylpyrrolidin-3-yl)methyl](methyl){[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
10-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
1-(5-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}thiophen-2-yl)ethan-1-one
1-(carbamoylmethyl)-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)piperidine-4-carboxamide
8-(2,3-dihydro-1H-inden-2-yl)-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-methyl-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N3-[(1R)-1-(4-methoxyphenyl)ethyl]-N5-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-benzoyl-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
1-(3,4-dimethoxybenzoyl)-N-(3,4-dimethylphenyl)piperidin-3-amine
N-[(1S,2R)-2-aminocyclobutyl]-2,3-dimethylquinoxaline-6-carboxamide
2-(pyridin-3-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)pyrimidine-5-carboxamide
2-[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]-4-(trifluoromethyl)pyrimidine
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-hydroxy-2-methylpropan-2-yl)acetamide
3-[5-(4-methylphenoxymethyl)-1,3,4-thiadiazol-2-yl]-1-[(2-methylpyridin-4-yl)methyl]urea
2-{3-hydroxy-5-[2-(piperidin-2-yl)ethyl]phenyl}benzoic acid
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)benzamide
{[3-(4-fluorophenyl)-1,2-oxazol-5-yl]methyl}[1-(1H-imidazol-1-yl)propan-2-yl]amine
N-methyl-3-[(oxolan-3-yl)sulfamoyl]-N-(1,3-thiazol-2-ylmethyl)benzamide
3-{1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl}-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-({5-fluoro-7-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1-benzofuran-2-carboxamide
2-[(5-{3-[(4-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)(ethyl)amino]ethan-1-ol
3-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1-{2-[2-(pyridin-2-yl)ethyl]phenyl}urea
3-({[(1-methyl-4-phenylpiperidin-4-yl)methyl]amino}methyl)piperidin-3-ol
13-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
N-(1-{1-[2-(3-chlorophenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
2-{3-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-ylmethyl]phenoxy}ethan-1-ol
2-(1-cyclohexyl-4-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperazin-2-yl)ethan-1-ol
5-(4-methanesulfonylphenyl)-2-methoxypyridine
3-methyl-4-[2-(3-methylphenyl)pyrimidin-5-yl]-4H,5H,6H,7H-[1,2]thiazolo[5,4-b]pyridin-6-one
4-(5-ethyl-1,3-oxazole-4-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
2-[1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
dimethyl(2-{[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]oxy}hex-5-en-1-yl)amine
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-3-(methylsulfanyl)propanamide
1-methyl-3-(2-methylpropyl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
N-[4-(3-fluorophenyl)phenyl]-1-(5-methylpyrazine-2-carbonyl)piperidine-3-carboxamide
3-({4-[3-(piperidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
(2S,4S)-1-(2,5-dimethylfuran-3-carbonyl)-N-ethyl-4-[2-(methylsulfanyl)acetamido]pyrrolidine-2-carboxamide
(4aS,8aR)-1-propyl-6-[4-(thiophen-2-yl)butanoyl]-decahydro-1,6-naphthyridin-2-one
(1S,4S)-2-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}-2-azabicyclo[2.2.1]heptane
1-[(2-chlorophenyl)methyl]-N-ethyl-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
6-(3-fluorophenyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}-3-({[2-(pyrrolidin-1-yl)ethyl]amino}methyl)piperidin-2-one
N-(pyrimidin-4-ylmethyl)-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
3-(2-methyl-1H-imidazol-1-yl)-1-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)propan-1-one
2-methyl-4-({3-[3-(1-methyl-1H-imidazol-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)-1,3-thiazole
1-[(2,3-difluorophenyl)methyl]-3-{1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl}-3-hydroxypiperidin-2-one
6-(3-acetylphenyl)-N,N-dimethylpyridine-2-carboxamide
7-{[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]methyl}-2-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one