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N-[2-methyl-1-(piperidin-1-yl)propan-2-yl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}morpholine-2-carboxylic acid
{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(pyrimidin-4-ylmethyl)amine
1-ethyl-4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-2-one
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(1-methylpyrrolidin-2-yl)ethyl]amine
2-(2-chloro-4-fluorophenyl)-N-[(1s,4s)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]acetamide
methyl 2-hydroxy-5-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}benzoate
5-(4-fluoro-2-methoxyphenyl)pyrazine-2-carboxylic acid
4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-dimethylpiperazine-1-sulfonamide
2-{[7-acetyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl](methyl)amino}-N-methylacetamide
2-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
(5R)-5-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)pyrrolidin-2-one
2-[methyl(pyridin-3-ylmethyl)amino]-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)acetamide
4-(2-methylpyridine-3-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
5-{1-[(1R)-1-(4-methoxyphenyl)ethyl]-1H-imidazol-2-yl}-2-(pyrrolidin-1-yl)pyrimidine
1-[benzyl(methyl)amino]-3-(2-methoxy-5-{[(pyridin-4-ylmethyl)amino]methyl}phenoxy)propan-2-ol
{[4-(benzyloxy)-3-methoxyphenyl]methyl}[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
2-methyl-3-(1H-pyrazol-1-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
1-(furan-2-ylmethyl)-4-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazine
N-(2,2-dimethyloxan-4-yl)-N-ethyl-2-propylpyridine-4-carboxamide
1-(1-benzofuran-2-ylmethyl)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]piperidine-3-carboxamide
4-[(3-fluorophenyl)methyl]-3-{2-[4-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
N4-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N4-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-(2-methylpropyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
methyl 4-[4-({4-[(4-fluorophenyl)methyl]-3-oxopiperazin-1-yl}methyl)-5-methyl-1,3-oxazol-2-yl]benzoate
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(3,5-dichloropyridin-4-yl)methyl]pyrrolidin-3-yl]methanol
N-methyl-N-[2-(oxan-4-yl)ethyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl}){[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}amine
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]pyrrolidin-3-yl]methanol
1-[9-(cyclopropylmethyl)-7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-(methylsulfanyl)ethan-1-one
naphthalen-1-yl (7S,9aR)-6,9-dioxo-7-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
7-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
7-fluoro-2-(1H-pyrazol-4-yl)-N-(1,1,1-trifluoropropan-2-yl)quinoline-4-carboxamide
1-{3-[3-(4H-1,2,4-triazol-4-yl)phenyl]benzoyl}piperidine
1-[4-(7-chloro-3-{[(2-phenylpropyl)amino]methyl}quinolin-2-yl)piperazin-1-yl]ethan-1-one
2-(4-methanesulfonylphenyl)-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]ethan-1-one
[1-(dimethyl-1,3-thiazol-4-yl)ethyl]({[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl})methylamine
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]acetamide
(2S,4R)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
5-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(3R,4S)-1-[5-(ethylsulfanyl)thiophene-2-carbonyl]-3,4-dimethylpiperidin-4-ol
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
2-[(1,1-dioxo-1λ6-thian-3-yl)methyl]benzonitrile
(1R,5S,6R)-3-(1-benzofuran-2-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
2-fluoro-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-5-sulfamoylbenzamide
3-[1-methyl-5-(5-methyl-1-phenyl-1H-pyrazol-4-yl)-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
2-methoxy-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethan-1-one
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(2-methylpropyl)-N-{2-[(pyridin-3-yl)amino]ethyl}-1,2-oxazole-5-carboxamide
7-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine