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5-ethyl-5-[1-(5-phenyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
6-methyl-N-[2-(4-phenylpyrimidin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-{4-[4-(adamantan-2-yl)piperazine-1-carbonyl]piperidin-1-yl}-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
2-amino-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]-5-methyl-6-(5-methylfuran-2-yl)pyridine-3-carbonitrile
2-[(5-{[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]methyl}pyrimidin-2-yl)(methyl)amino]acetic acid
3-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-1,2-dihydroquinoxalin-2-one
7-(6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydro-2H-1-benzopyran-2-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[(4-phenyl-1,3-thiazol-2-yl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-methyl-3-(2-methylpropyl)-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-1H-pyrazole-5-carboxamide
1-methyl-3-{2-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)urea
N-ethyl-5-{4-[(methylsulfanyl)methyl]piperidine-1-carbonyl}pyrimidin-2-amine
2-cyclopropyl-N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,3-benzoxazole-6-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
(3S,4R)-1-(5-fluoro-2-methoxybenzoyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
3-(1H-1,2,3-benzotriazol-1-yl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
4-(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidine-3-carbonyl)morpholine
N-(2-{7-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-[1-(5-{[benzyl(methyl)amino]methyl}-1,2-oxazole-3-carbonyl)piperidin-2-yl]ethan-1-ol
3-[4-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-1-yl]propanamide
1-methyl-4-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4-phenylpiperidine
2-benzyl-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1,3-thiazole-4-carboxamide
3-tert-butyl-1-methyl-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(2-aminoethyl)-N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}quinazolin-4-amine
6-(2-hydroxyethyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-({[1-(1,3-thiazol-4-ylmethyl)piperidin-3-yl]oxy}methyl)pyridine
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-6-methyl-2-(4-methylphenoxymethyl)-1-[2-(morpholin-4-yl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{4-[2-(2-methoxyethyl)morpholin-4-yl]quinazolin-2-yl}ethan-1-amine
N-methyl-2-(2-methylpropyl)-4-oxo-N-phenyl-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxamide
4-(5-methoxypyridin-3-yl)-1H-indole
2-(4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-N-ethylacetamide
2-(4-{[({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenoxy)ethan-1-ol
3-{3-[5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-(piperidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-1-yl]propyl}pyridine
4-{1-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H-imidazol-2-yl}benzoic acid
(1S,5R)-3-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-3,9-diazabicyclo[3.3.2]decan-10-one
(2S,4S)-4-amino-1-[2,4-bis(trifluoromethyl)benzoyl]-N-methylpyrrolidine-2-carboxamide
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-methyl-N-(quinoxalin-6-ylmethyl)propanamide
5-(2,3-difluoro-4-methoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
6-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methoxyphenyl]-N,N-dimethylpyridine-3-carboxamide
(3S,4S)-1-(2,1,3-benzothiadiazole-4-sulfonyl)piperidine-3,4-diol
1-(4-chloro-3-methylbenzoyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N-tert-butyl-N'-methyl-N'-[1-(3-phenylpropyl)piperidin-3-yl]ethanediamide
1-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(oxolan-3-yl)benzamide
5-{[2,2-bis(prop-2-en-1-yl)piperidin-1-yl]methyl}-N-ethylpyrimidin-2-amine
N-{2-[3-(2-methylpropyl)-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl]ethyl}acetamide
N-({3-methyl-7-[2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-2-yl)acetamide