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(2S,4S,5R)-2-ethyl-4-[(furan-3-ylmethyl)carbamoyl]-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
3-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-ethoxybenzoic acid
9-ethyl-4-[5-(methoxymethyl)thiophene-2-carbonyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-3-(1H-imidazol-1-yl)propan-1-one
1-(3-chloro-4-methoxyphenyl)-3-(2,2-dimethyloxan-4-yl)-3-ethylurea
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]butanamide
(3S,4R)-4-phenyl-1-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
8-[(2-chloro-4,5-diethoxyphenyl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-methyl-4-{[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]methyl}benzamide
3-phenyl-N-{1-[1-(pyridine-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-yl}ethan-1-ol
1-{2-[2-(2,4-dichlorophenyl)-1H-imidazol-1-yl]propyl}-1H-1,2,4-triazole
N-(2,6-dimethoxypyridin-3-yl)-4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidine-1-carboxamide
N-({7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-(3-fluorophenyl)acetamide
(2E)-3-(1H-imidazol-4-yl)-1-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]prop-2-en-1-one
{1-[1-(adamantane-1-carbonyl)piperidin-4-yl]-2-phenylethyl}(methyl)(pyridin-3-ylmethyl)amine
2-cyclohexyl-N-{5-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl}acetamide
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-phenyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-[3-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}azetidin-3-yl)pyridine
N-(4-{4-[(2,2-dimethyloxan-4-yl)amino]piperidin-1-yl}phenyl)-2H-1,3-benzodioxole-5-carboxamide
2-chloro-N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-5-(trifluoromethyl)benzamide
N-ethyl-3-{9-oxo-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-2-yl}propanamide
4-[(2-fluorophenyl)methyl]-3-{2-oxo-2-[4-(pyrrolidin-1-yl)piperidin-1-yl]ethyl}piperazin-2-one
2-[(4-methyl-1-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-1,3-benzodiazol-2-yl)methoxy]acetic acid
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylpropyl)acetamide
(3S,5S)-5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-1-methylpyrrolidin-3-amine
ethyl 2-{5-[1-(cyclooctylamino)ethyl]-4H-1,2,4-triazol-3-yl}acetate
4-(4-chlorophenyl)-N-[1-(4-methylphenyl)-5-oxopyrrolidin-3-yl]butanamide
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylsulfanyl)benzamide
1-(1-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1,4-diazepan-5-one
1-{4-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]thiophen-2-yl}ethan-1-one
4-methyl-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]quinoline
3-(2-methoxybenzoyl)-1-phenylmethanesulfonylpiperidine
1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidine-4-carboxamide
1-(2-methylphenyl)-3-(1-{1-[1-(4-methylpyridin-2-yl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
N,N-diethyl-1-({1-[(3-fluorophenyl)methyl]-6-methyl-2-oxo-1,2-dihydroquinolin-3-yl}methyl)piperidine-3-carboxamide
5-[2-(1-cyclohexyl-3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]-4,6-dimethylpyrimidin-2-ol
(2S)-2-[(2-amino-5-methylpyrimidin-4-yl)amino]-3-cyclohexylpropan-1-ol
1-(4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)isoquinoline
(1R,5R)-3-methanesulfonyl-6-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(5S,9aS,9bS)-2-phenyl-5-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]hexan-1-one
methyl (1R,5S,6R)-6-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}-3-azabicyclo[3.1.0]hexane-3-carboxylate
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-4-[(3-fluorophenyl)methyl]-1,4-diazepane
2-amino-N-[1-(3-fluorophenyl)-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]acetamide
N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-(methoxymethyl)-1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
N,N,5-trimethyl-2-[4-(2-propoxyethyl)piperazin-1-yl]pyrimidin-4-amine
3-{[2-(4-cyclohexyl-1,4-diazepan-1-yl)pyrimidin-4-yl](methyl)amino}propane-1,2-diol