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(3S,4S)-N-benzyl-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidine-1-sulfonamide
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyrazolo[1,5-a]pyridine-7-carboxamide
1-{[3-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1H-pyrazol-5-yl]methyl}-1H-1,3-benzodiazole
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-5-phenylpentanamide
2,6-dimethoxy-N-[4-(2-methoxyphenyl)-1,3-dimethyl-1H-pyrazol-5-yl]benzamide
4-(4-methyl-1H-pyrazol-3-yl)-N-[3-(1,3-oxazol-5-yl)phenyl]piperidine-1-carboxamide
N,N-dimethyl-3-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]piperidine-1-carboxamide
1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-3-phenylpiperazine
N-cyclopentyl-2-methoxy-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}acetamide
9-(4-methoxybenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-(naphthalene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-fluoro-3-methyl-2-[4-phenyl-1-(1H-1,2,4-triazol-5-ylmethyl)-1H-imidazol-5-yl]-1H-indole
[3-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)piperidin-3-yl]methanol
3-{methyl[(4-methylphenyl)methyl]sulfamoyl}-N-[(2S)-pyrrolidin-2-ylmethyl]benzamide
(4aS,7aR)-1-[2-(4-methylphenoxy)acetyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-{1-[2-(5-methylfuran-2-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}phenoxy)ethan-1-ol
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
ethyl 4-({[2-methyl-3-(1H-pyrrol-1-yl)phenyl]carbamoyl}amino)piperidine-1-carboxylate
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
7-(pyridin-3-ylmethyl)-2-[3-(thiophen-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
4-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl)-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
3-(benzyloxy)-1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidine
[(4-{1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-2-yl}phenyl)methyl]dimethylamine
2-oxo-N-phenyl-2-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}acetamide
(1R,5S,6R)-3-cyclopentyl-N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-3-(4-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-[2-methoxy-5-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
4-(3-fluorophenoxy)-1-(4-methyl-1H-imidazole-5-carbonyl)piperidine-4-carboxylic acid
1-{[1-(ethoxymethyl)cyclobutyl]methyl}-5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazole
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
2-({2-[1-(2-methoxy-6-methylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
2-(1H-indol-1-yl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-[4-({[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amino}methyl)thiophen-2-yl]ethan-1-one
(3S,4S)-3-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-4-hydroxy-1λ6-thiolane-1,1-dione
5-methyl-4-[1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-2-[(pyridin-2-ylmethyl)sulfanyl]pyrimidine
N-methyl-N-[2-(4-methylphenoxy)ethyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
5-fluoro-N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}quinazolin-4-amine
N'-(2-methoxyethyl)-N-(4-methyl-1,3-thiazol-2-yl)-N'-(thiophen-2-ylmethyl)ethanediamide
6-methyl-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3,4-dihydroquinazolin-4-one
1-{1-[1-(2,6-dimethoxybenzoyl)piperidin-4-yl]ethyl}-4-methylpiperazine
N-[(2-propyl-1,3-thiazol-4-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
1-[4-({3-[3-(azepan-1-yl)-2-hydroxypropoxy]phenyl}methyl)piperazin-1-yl]ethan-1-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[(oxan-3-ylmethyl)amino]pyridine-3-carboxamide
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamide
6-fluoro-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-1,3-benzodiazole-2-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetamide
8-methoxy-N-(thian-4-yl)-3,4-dihydro-2H-1-benzopyran-3-amine
1-(2-{[2-(1H-imidazol-2-yl)ethyl]amino}pyrimidin-4-yl)piperidin-4-ol