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(3S,4R)-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-amino-4-(4-methanesulfonylphenyl)-6-(3-methoxyphenyl)pyridine-3-carbonitrile
N2-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]pyrimidine-2,4-diamine
2-(2H-1,2,3-benzotriazol-2-yl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]acetamide
2-{4-[2-methyl-2-(morpholin-4-yl)propyl]piperazin-1-yl}pyridine-3-carboxamide
2-amino-6-(1,3-dimethyl-1H-pyrazol-4-yl)-4-[4-methoxy-3-(methoxymethyl)phenyl]pyridine-3-carbonitrile
1-(2-cyclohexylethyl)-3-hydroxy-3-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)piperidin-2-one
(3S,4R)-N,N-dimethyl-1-(5-methyl-1,2-oxazole-3-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-amine
N-methyl-2-(1-oxo-1,2-dihydroisoquinolin-2-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
N-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
2-({2-[2-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
1-tert-butyl-2-(4,4,4-trifluorobutyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
1-(4-benzylpiperazin-1-yl)-3-{1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidin-3-yl}propan-1-one
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](methyl){[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-{2-[(4-butylphenyl)carbamoyl]ethyl}piperidine-4-carboxamide
5-[3-(furan-2-amido)-2-methylbenzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
methyl 4-{[3-(2-{[(3-methoxyphenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]methyl}benzoate
4-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1-oxaspiro[4.4]nonan-2-one
1-methyl-N-[(1-methylpiperidin-2-yl)methyl]-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)[(2,3,4-trimethoxyphenyl)methyl]amine
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
ethyl 4-[2-(methoxymethyl)-1-methyl-5-(2-phenylacetamido)-1H-1,3-benzodiazole-7-carbonyl]piperazine-1-carboxylate
1-(3-methoxyphenyl)-6-methyl-4-[2-(2-oxo-4-phenylpyrrolidin-1-yl)acetyl]piperazin-2-one
[(3R,4R)-1-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
5,6-dimethyl-N-(oxolan-2-ylmethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]pyridine-3-carboxamide
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[2-(2,5-dimethylphenoxy)ethyl]-N-methylacetamide
1-benzyl-5-{[(5-fluoro-2-methylphenyl)methyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{2-[1-(pyrrolidine-1-carbonyl)piperidin-2-yl]ethyl}phenol
N-(dicyclopropylmethyl)-6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
{[4-(1H-imidazol-1-yl)phenyl]methyl}(methyl)(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
[(8-methoxy-2H-chromen-3-yl)methyl](methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
2-(3-methylbutyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[3-(dimethylamino)-2,2-dimethylpropyl]-1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N,N-dimethyl-2-[(4-phenylbutan-2-yl)amino]ethane-1-sulfonamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]piperidine-3-carboxamide
N-benzyl-2-{4-[1-(carbamoylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}acetamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-4-(pyrrolidin-1-ylmethyl)benzamide
{[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl}[(2-methoxyphenyl)methyl]amine
N-{[1-(dimethylamino)cyclohexyl]methyl}-2-oxo-1-phenylpyrrolidine-3-carboxamide
N-cyclopropyl-N-(3-phenylprop-2-yn-1-yl)-3-propanamidobenzamide
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(thiophen-3-ylmethyl)piperazine
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-4-yl)propanamide
5-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-4-(propan-2-yl)-1,2,3-thiadiazole
5-methyl-5-{1-[6-(propan-2-yl)pyridazin-3-yl]piperidin-4-yl}imidazolidine-2,4-dione
1-(2-ethoxyethyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
4-(4-methyl-1H-pyrazol-1-yl)-1-[(6-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidine-4-carboxylic acid
4-[(dipropylamino)methyl]-N-(4-hydroxybutyl)benzamide
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(furan-2-ylmethyl)acetamide
N-{2-methyl-4-[2-(morpholin-4-ylmethyl)phenyl]phenyl}pyridine-3-carboxamide