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1-[2-(4-hydroxypiperidin-1-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one
N-(cyclohexylmethyl)-2-{2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}acetamide
2-({[2-chloro-5-(morpholine-4-carbonyl)phenyl]carbamoyl}amino)acetamide
2-chloro-5-{[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyridine
2-chloro-4-(3-cyano-4,5,6-trimethylpyridin-2-yl)benzamide
N-cyclopentyl-2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propanamide
N5-cycloheptyl-1-cyclopropyl-N3-methyl-4-oxo-N3-(quinolin-5-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
4-(3-chloropyridin-2-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
5-methyl-3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-{4-chloro-3-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]phenyl}acetamide
N-[2-(1,4-dioxo-1,2,3,4-tetrahydrophthalazin-2-yl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
1-ethyl-3-methyl-8-[1-(methylsulfanyl)propan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}acetamide
(2S,4R)-N-ethyl-1-(furan-2-carbonyl)-4-[3-(1H-pyrrol-1-yl)propanamido]pyrrolidine-2-carboxamide
5-chloro-3-ethyl-4-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-1-methyl-1H-pyrazole
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-(methoxymethyl)-N-(quinolin-3-ylmethyl)-1H-pyrazole-4-carboxamide
2-phenyl-N-{[7-(quinolin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}acetamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(thiophen-2-yl)propan-1-one
N-({1-[(2-ethylpyrimidin-4-yl)methyl]pyrrolidin-3-yl}methyl)-6-methylpyridine-3-carboxamide
3-(pyrrolidine-1-carbonyl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]benzene-1-sulfonamide
3-methoxy-N-{1-[(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)methyl]-1H-pyrazol-5-yl}benzamide
N-({5-[(2-cyanophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
methyl (2S,4S)-4-(2,6-dichlorobenzamido)-1-methylpyrrolidine-2-carboxylate
N-{2-cyclobutyl-1-methyl-7-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
5-ethyl-N4-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidine-2,4-diamine
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-hydroxy-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
(1R,5R)-3-cyclobutanecarbonyl-6-[(3,4-dimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(2H-1,3-benzodioxol-5-yl)piperidin-4-amine
1-{4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-[(3S,4R)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
5-{3-[(benzyloxy)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-4-methyl-1,3-thiazole
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
3-(2-methylquinolin-5-yl)-1-(oxolan-2-ylmethyl)-1-(pyridin-2-ylmethyl)urea
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
2-(1-benzyl-4-phenylpiperidine-4-carbonyl)-1,2-oxazolidin-4-ol
4-[(8-methoxyquinolin-2-yl)methyl]-5-methyl-1-(2-methylphenyl)piperazin-2-one
(1S,5R)-6-[(2,6-difluorophenyl)methyl]-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-[3-(benzylsulfanyl)propanoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-methyl-N-[2-phenyl-1-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)ethyl]thiophene-2-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]-4-methyl-1H-imidazole-2-carboxamide
1-(1H-1,2,3-benzotriazole-5-carbonyl)-N-(3,4-dimethylphenyl)piperidin-3-amine
4-({2-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]phenyl}methyl)morpholine
1-{4-[(3R)-3-hydroxypyrrolidin-1-yl]-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one
N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
N-cyclopentyl-N'-[3-(2-methoxybenzamido)phenyl]ethanediamide
methyl 2-[2-(2,1,3-benzoxadiazol-4-yl)-1H-imidazol-1-yl]-4-(methylsulfanyl)butanoate
3-benzyl-5-[(3-cyclohexylpyrrolidin-1-yl)methyl]-1,2,4-oxadiazole
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-ethylbutan-1-one
2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]benzamide