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1-[4-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
5-cyclopentyl-1-(2-hydroxyethyl)-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-fluoro-2-[1-(morpholine-4-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
N-[(3,4-dimethoxyphenyl)methyl]-4-phenyl-N-(pyridin-3-ylmethyl)benzamide
N-(furan-2-ylmethyl)-2-(morpholin-4-yl)-N-(prop-2-yn-1-yl)benzamide
ethyl 1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylate
1-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(propan-2-yloxy)ethan-1-one
6-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1H-indole
5-(cyclohexylamino)-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-(cyclopropylmethyl)-2-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
4-acetamido-N-[2-(1-hydroxycyclopentyl)ethyl]-N,2-dimethylbenzamide
methyl 2-[4-(4-methyl-1,4-diazepan-1-yl)-6-oxo-1,6-dihydropyridazin-1-yl]hexanoate
{1-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-3-yl}methanol
1-({3-[(4,6-dimethylpyridin-2-yl)carbamoyl]phenyl}methyl)piperidine-3-carboxamide
(2S,4R)-4-amino-N-(propan-2-yl)-1-(5-propylthiophene-3-carbonyl)pyrrolidine-2-carboxamide
N-[(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
2,2-dimethyl-N-({1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-3-yl}methyl)propanamide
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(morpholin-4-yl)ethan-1-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
2-{5-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidin-5-yl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
6-[(1-phenylethyl)sulfamoyl]-N-(propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-[5-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-[(4-methoxyphenyl)methyl]-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
1'-[3-(4-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-{2-[2-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidine-2,5-dione
1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]urea
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(2-phenylethyl)pyrrolidin-3-yl]-5-methyl-1,2-oxazole-3-carboxamide
N-[3-(cyclopentyloxy)phenyl]-8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
1-{[1-(4-hydroxy-3-methylbenzoyl)piperidin-4-yl]methyl}pyrrolidin-2-one
N-butyl-N-methyl-3-{[methyl(oxolan-2-ylmethyl)amino]methyl}imidazo[1,2-a]pyridine-2-carboxamide
1-(cyclopropylmethyl)-5-(2-fluorophenyl)-1H,4H-pyrazolo[3,4-d]imidazole
7-(cyclohexylmethyl)-2-[3-(1H-pyrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one
(3S,9aR)-3-[(1R)-1-hydroxyethyl]-8-[(3-methylthiophen-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[(4-fluorophenyl)methyl]-1-(oxolan-3-ylmethyl)piperidine
N-(2,3-dihydro-1H-inden-1-yl)-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
2-{methyl[(2E)-3-phenylprop-2-en-1-yl]amino}-N-(1,3-thiazol-2-yl)propanamide
3-[2-(3-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5,6-dimethoxy-2-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1,2-dihydroisoquinolin-1-one
N-[(4-fluorophenyl)methyl]-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
8-[4-(propan-2-yl)benzoyl]-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
N-butyl-N-[(5-methylthiophen-2-yl)methyl]-2-(1H-1,2,4-triazol-5-yl)benzamide
5-(3,4,5-trimethoxyphenyl)pyrazin-2-amine
(3S,4S)-1-(7-methoxy-4-methylquinazolin-2-yl)-4-(piperidin-1-yl)pyrrolidin-3-ol
1-{2-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
N-[4-({[1-(pyrazin-2-yl)propan-2-yl]carbamoyl}methyl)phenyl]butanamide
2-(1,3-benzoxazol-2-ylsulfanyl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]butan-1-one
2-(2-{7-[cyclohexyl(methoxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-oxoethyl)-4-methyl-1,2-dihydrophthalazin-1-one
5-[5-(ethanesulfonyl)thiophen-2-yl]-1,2,3,4-tetrahydroisoquinoline