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2-[(3,4-difluorophenyl)methyl]-8-(6-methylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
(4aS,7aR)-1-(4-ethylbenzoyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(4-methylphenoxy)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}acetamide
4,6-dimethyl-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
3-ethyl-1-({1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)urea
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(2-hydroxyethyl)propanamide
2-methyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-3-[(pyridin-2-ylmethyl)amino]benzamide
N-(furan-2-ylmethyl)-N-methyl-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide
2-{4-[4-fluoro-3-(hydroxymethyl)phenyl]phenyl}-N-methylacetamide
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
8-chloro-2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}quinoline
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-8-fluoroquinoline-2-carboxamide
7-{3H-benzo[e]indole-2-carbonyl}-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[3-(furan-2-amido)-4-methoxyphenyl]-4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
(3S,5R)-N3-(6-methylpyridin-3-yl)-N5-[2-(pyrazin-2-yl)ethyl]piperidine-3,5-dicarboxamide
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(1-methoxybutan-2-yl)pyridin-2-amine
N'-(2-ethoxyphenyl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}propanediamide
3-({6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-1,3-oxazolidin-2-one
N-(3-acetamido-4-fluorophenyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carboxamide
N-cyclopropyl-3-[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]propanamide
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]methanol
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-4-({[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2-methylpyrrolidin-2-yl]methanol
N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1H-pyrazole-5-carboxamide
N,N-diethyl-1-(1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-amine
3-(3,5-dimethylphenyl)-N-[(4-methanesulfonylmorpholin-2-yl)methyl]propanamide
2-[4-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)piperazin-1-yl]pyridine-3-carbonitrile
N-[(3-chlorophenyl)methyl]-3-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]propanamide
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(oxolan-2-ylmethyl)benzamide
9-[(4-ethylphenyl)methyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(azepane-1-carbonyl)-7,8-dimethyl-2-(2-methylpyrimidin-5-yl)quinoline
4-{5-[3-(furan-2-yl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-1H-pyrazole
N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-(2-methoxyethyl)-2,3-dihydro-1H-indene-2-carboxamide
N-[(4-phenyloxan-4-yl)methyl]-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-{[3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
5-{2-[4-phenyl-5-(1,3-thiazol-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
(2S,4S)-4-amino-N-ethyl-1-[(5-methyl-2,1,3-benzothiadiazol-4-yl)sulfonyl]pyrrolidine-2-carboxamide
N-(1-hydroxypropan-2-yl)-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
N-methyl-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-N-[1-(pyrimidin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
2-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
N-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)-4-methyl-1,2,3-thiadiazole-5-carboxamide
6-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
4-{3-[(4S,4aS,8aR)-4-hydroxy-4-phenyl-decahydroquinoline-1-carbonyl]piperidin-1-yl}-2-(2-methoxy-2-methylpropyl)-2,3-dihydro-1H-isoindole-1,3-dione
4-cyclobutyl-N-(1,4-dioxan-2-ylmethyl)-6-methylpyrimidin-2-amine
methyl 3-[(2-methylphenyl)methyl]-9-[(1-methylpiperidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(3S,4R)-1-(2-hydroxypyridine-3-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
1-(1-{3-[4-(difluoromethoxy)phenyl]phenyl}ethyl)pyrrolidine
(3-{2-[1-(2,3-difluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
5-(2,6-dimethoxyphenyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2,4-triazin-3-amine
2-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)pyrimidine