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(4aS,7aR)-1-(1,5-dimethyl-1H-indazole-3-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,N,2-trimethyl-7-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
8-[(3-fluoro-2-methylphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(2H-1,3-benzodioxol-5-yl)-N-(1-butyl-4-methyl-1H-pyrazol-5-yl)propanamide
(3aS,6aR)-5-(5-ethyl-2-methylpyrimidin-4-yl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(dimethyl-1,3-thiazol-2-yl)pyrrolidin-3-yl]methanol
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(1-methyl-1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2-methyl-1-benzofuran-7-carboxamide
8-(5,6-dimethylpyrimidin-4-yl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
1-(1-benzofuran-2-ylmethyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-(2-hydroxyethyl)-3-(5-{thieno[2,3-d]pyrimidin-4-yl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanamide
4-{[3-(heptan-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]sulfonyl}morpholine
8-(1-benzofuran-2-ylmethyl)-1-ethyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(furan-2-yl)phenyl]-3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carboxamide
1-(furan-2-carbonyl)-4-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,4-diazepane
N-{3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propyl}pyrimidin-4-amine
N-[3-(1H-imidazol-1-yl)propyl]-4-(4-methylphenoxy)piperidine-4-carboxamide
4-{3-cyclopropyl-5-[2-phenyl-1-(1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}-2-methylpyridine
1-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-[4-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]pyridazine-3-carboxamide
N-{[3-methyl-7-(3-phenoxypropanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(pyrimidin-2-ylsulfanyl)acetamide
2-{[3-(propan-2-yloxy)phenyl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-tert-butyl-2-({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)acetamide
5-ethyl-6-methyl-N4-[(5-methyl-1H-pyrazol-3-yl)methyl]pyrimidine-2,4-diamine
2-methyl-8-[6-methyl-2-(methylsulfanyl)pyrimidin-4-yl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(3S,4R)-4-methyl-1-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]piperidine-3,4-diol
4-(2-phenylethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-({4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}methyl)pyridin-2-amine
N-[1-(7-{[4-(dimethylamino)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-2-methylpropyl]propanamide
3-{1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
(3R,5S)-N-cyclohexyl-1-[(1-methyl-1H-imidazol-2-yl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
2-[1-(propan-2-yl)piperidin-4-yl]-1-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-yl)ethan-1-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[3-(1H-pyrrol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
(3S,4S)-1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
7-cyclohexyl-2-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(1R,5R)-6-[(2-chloro-6-fluorophenyl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(4-methanesulfonylphenyl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
(3S,4S)-4-methyl-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidine-3,4-diol
2-[3-({4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}methyl)phenoxy]acetamide
3-({ethyl[2-(morpholin-4-yl)ethyl]amino}methyl)-6-methyl-1,2-dihydroquinolin-2-one
1-{1-[6-(azocan-1-yl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
1-[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]piperidine-3-carboxamide
(1S,5R)-6-[2-(methylsulfanyl)pyridine-3-carbonyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
7-[(4-fluorophenyl)methyl]-2-[(2E)-2-methylbut-2-en-1-yl]-2,7-diazaspiro[4.5]decan-6-one
methyl (2S)-1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidine-2-carboxylate
4-acetyl-N-[4-(3-methoxyphenoxy)phenyl]-1,4-diazepane-1-carboxamide
1-(3-methylpyridin-4-yl)-4-[4-(pyridin-3-yl)pyrimidin-2-yl]-1,4-diazepane
2-(4-oxo-1,4-dihydroquinolin-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
8-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)quinoline
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)furan-2-carboxamide