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1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-{4-[(2-aminopyridin-3-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
4-{4-[1-(4-chlorophenyl)cyclopropanecarbonyl]piperazin-1-yl}-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-[(2,3-dichloro-6-fluorophenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}){[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl}amine
6-{[(2,3-dimethyl-1H-indol-5-yl)methyl]amino}pyridine-3-carbonitrile
1-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)-4-(2-methoxyphenyl)piperazine
1-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)(pyridin-4-ylmethyl)amine
2-(4-fluorophenyl)-1-[3-(3-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]ethan-1-one
N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
2,3-dimethyl-6-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanoyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-[4-methyl-4-(methylsulfanyl)pentan-2-yl]-1-(pyridin-3-ylmethyl)piperidin-4-amine
N'-(2-fluoro-5-methylphenyl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}butanediamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-[methyl(phenyl)amino]acetamide
2-[5-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}acetamide
N-tert-butyl-2-({[1-(2-cyclohexylethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}amino)acetamide
1-(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-3-methylbutan-1-ol
3-{[4-(hydroxymethyl)oxan-4-yl]methyl}-3-methyl-1-[4-(2-methylphenyl)phenyl]urea
N-{3-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyridin-3-amine
4-{[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
1-(3,5-dimethylphenyl)-4-{2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}piperazin-2-one
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(3-methylbut-2-en-1-yl)piperidine-4-carboxamide
8-(2-amino-2-methylpropanoyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 3-(2-hydroxyethyl)-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(2-chloropyridin-3-yl)-3-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}urea
6-(3-fluorophenyl)-N-(3-hydroxy-2,2-dimethylpropyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-[(1,2-oxazol-3-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
1-{6-[3-(1H-pyrazol-1-yl)phenyl]pyridin-2-yl}ethan-1-ol
4-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}-1λ6-thiomorpholine-1,1-dione
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-8-methoxyquinoline
6-[(oxan-4-ylmethyl)amino]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
methyl[(3-methyl-1H-indol-2-yl)methyl]{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}furan-2-carboxamide
3-chloro-N-(2-methoxyethyl)-4-({1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}oxy)benzamide
2-({4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)-5-methoxyphenol
N-(4-methylphenyl)-2-oxo-2-{2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-yl}acetamide
N-{imidazo[1,2-a]pyrazin-3-ylmethyl}-3-(pyridin-3-yl)propanamide
2-{[1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]formamido}-N-(propan-2-yl)acetamide
4-methyl-2-[4-(oxolan-3-ylmethyl)piperazin-1-yl]-6-(trifluoromethyl)pyrimidine
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)[(2-methyl-1,3-oxazol-4-yl)methyl]amine
1-(5-methoxy-2-{[methyl(pyrimidin-4-ylmethyl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1,3-thiazole-4-carboxamide
[(2-chlorophenyl)methyl]({[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl})amine
N-{1-[({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}pyridine-2-carboxamide
4-fluoro-N-{[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}aniline
8-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
5-{1-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-2-ethylpyrimidine