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N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(2,3,4-trimethoxyphenyl)benzonitrile
2-{1-[(3,4-difluorophenyl)methyl]-4-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1-methylazepane-2-carboxamide
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
N-[(2R,3R)-2-ethoxy-1'-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
N-(1-{3-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)-2-methoxyacetamide
N'-cyclooctyl-N-methyl-N-[2-(oxan-4-yl)ethyl]butanediamide
N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-ethoxy-N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)acetamide
2-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}formamido)-N,N-dimethylpropanamide
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-[2-(2-hydroxyethoxy)ethyl]propanamide
2-(4-chlorophenyl)-N-[2-(4,5-dimethyl-1H-imidazol-1-yl)ethyl]-2-hydroxyacetamide
1-[2-(5-methylfuran-2-yl)phenyl]-3-[2-(pyrrolidin-1-yl)ethyl]urea
N-[3-(3-fluorophenyl)phenyl]-1-(pyrrolidine-1-carbonyl)piperidine-4-carboxamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(thiophene-2-carbonyl)pyrrolidin-3-yl]acetamide
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-{[2-(4-acetylpiperazin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-3-(2-methoxyphenyl)-N-(oxolan-2-ylmethyl)propanamide
N4-[(5-fluoro-2,3-dimethyl-1H-indol-7-yl)methyl]-6-methylpyrimidine-2,4-diamine
3-{1-[(2-chloro-6-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}-N,N-dimethylpiperidine-1-carboxamide
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
8-[(furan-2-ylmethyl)carbamoyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[({[4-(3-chlorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]phenol
2-({3-[benzyl(2-hydroxyethyl)carbamoyl]phenyl}amino)acetic acid
N-[3-(furan-2-yl)-3-phenylpropyl]-2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carboxamide
4-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
4-benzoyl-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidine
4-{1-[1-(2,5-dimethylpyrimidin-4-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
6-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)-1,4-oxazepan-6-ol
(2S,4S)-1-[(2E)-3-phenylprop-2-en-1-yl]-N-(propan-2-yl)-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
1-[2-({[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
1,4-dimethyl-2-(2-{8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}ethyl)piperazine
5-(1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
2-methyl-4-(3-{4-[2-(methylsulfanyl)ethyl]piperazine-1-carbonyl}phenyl)butan-2-ol
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
4-chloro-1-ethyl-N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-1H-pyrazole-5-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[2-(methylsulfanyl)pyrimidin-4-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-ethyl-3-(6-methyl-9H-purin-9-yl)benzamide
2-{3-[4-(3-chlorophenyl)piperazin-1-yl]propyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(ethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
2-methoxy-6-({[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenol
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-fluorobenzamide
1-(2H-1,3-benzodioxol-5-yl)-3-(2-phenylethyl)-5-(1H-1,2,4-triazol-5-yl)-1H-1,2,4-triazole
2-(4-{[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
5-tert-butyl-4-{[6-oxo-4-(piperazin-1-yl)-1,6-dihydropyridazin-1-yl]methyl}furan-2-carboxamide
1-[4-({[(4-chlorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-cyclopropyl-1-(2-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
ethyl 4-(3-{[(thiophen-2-ylmethyl)amino]methyl}-6H,7H,8H-cyclopenta[g]quinolin-2-yl)piperazine-1-carboxylate
7-(cyclopropylmethyl)-2-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one