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1-benzyl-8-(2,2-diphenylethyl)-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
(1R,5R)-N-(3-methoxy-4-methylphenyl)-3-azabicyclo[3.3.1]nonane-3-carboxamide
7-(3-chlorophenyl)-4-(pyridin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
2-[1-(2-methoxyphenyl)-5-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl]acetamide
6-cyclobutyl-2-(3-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenyl)-3,4-dihydropyrimidin-4-one
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-5-[(3-hydroxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(1S,5R)-6-methyl-3-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-propanoylpiperidine-3-carboxamide
{2-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}urea
3-phenyl-1-(5-propyl-1,3,4-oxadiazole-2-carbonyl)piperazine
5-methyl-N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-phenyl-1,2-oxazole-4-carboxamide
N-methyl-N-{1-[2-(2-oxo-1,2,3,4-tetrahydroquinolin-1-yl)acetyl]pyrrolidin-3-yl}acetamide
2-{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1,3-benzoxazole
1-(4-fluorophenyl)-4-[2-(1H-pyrazol-1-yl)benzoyl]-1,4-diazepane
1-[cyclohexyl(methyl)amino]-3-{2-[(cyclopentylamino)methyl]phenoxy}propan-2-ol
1-[6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
(4aR,7aS)-1-(4-methylpentanoyl)-4-(pyridazine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(2S)-1-{5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-2-yl]methanol
3-[2-(3-fluorophenyl)piperidine-1-carbonyl]-2-methoxypyridine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
(2-oxo-2-{9-oxo-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-2-yl}ethyl)urea
4-(2-{5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}ethyl)morpholine
1-[4-(4-fluorophenyl)-4-hydroxypiperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
8-methoxy-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
3-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
1-[2-(4-chlorophenyl)ethyl]-6-oxo-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
N-benzyl-1-(3-fluoro-4-methoxybenzoyl)-N-methylpiperidin-3-amine
8-methoxy-N-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
1,6-dimethyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1H-indole-2-carboxamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-N,N-dimethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
4-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-1,2,3-triazole
5-[6-(trifluoromethyl)pyridin-2-yl]pyrimidine
4-({[(2-chloropyridin-3-yl)methyl](methyl)amino}methyl)-2-fluoro-6-methoxyphenol
4-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidine
1-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-3-(1-propyl-1H-pyrazol-5-yl)urea
3-{[2-(cyclopropylmethyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]methyl}-1,2-dihydroquinolin-2-one
5-(2-methoxynaphthalen-1-yl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
6-(1H-pyrazol-3-yl)-2-(pyrrolidin-1-yl)pyrimidin-4-amine
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
1-benzyl-3-(2-methylpropyl)-8-[1-(methylsulfanyl)propan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4S)-1-(cyclohexylmethyl)-N-ethyl-4-(5-methoxyfuran-2-amido)pyrrolidine-2-carboxamide
(1R,3S)-3-methoxy-7-[4-(trifluoromethyl)pyridin-2-yl]-7-azaspiro[3.5]nonan-1-ol
1-methyl-3-(2-oxo-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}ethyl)imidazolidine-2,4-dione
[(5-{1-[(3,5-dichloropyridin-4-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
N-[(3R,4S)-1-cyclopentyl-4-cyclopropylpyrrolidin-3-yl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
3-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-phenylurea