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2,5-dimethyl-N-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}morpholine
2-[({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]pyridine-3-carboxamide
4-(2,6,8-trimethylquinoline-4-amido)oxane-4-carboxylic acid
methyl 5-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-[4-(trifluoromethyl)benzoyl]pyrrolidin-3-yl]methyl})amino]ethan-1-ol
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]acetamide
6-methyl-2-oxo-5-[6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-1,2-dihydropyridine-3-carbonitrile
2-{4-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-cyclohexylpiperazin-2-yl}ethan-1-ol
1-(azocan-1-yl)-3-[4-({[(2,5-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
N,2-dimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
3-({[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)propane-1,2-diol
4-{4-[({1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}amino)methyl]phenyl}but-3-yn-1-ol
7-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-2,7-diazaspiro[4.5]decane
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[1-(propan-2-yl)cyclopropyl]amino}methyl)piperidin-2-one
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-{[2-(methylsulfanyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
[(3-{[1-(furan-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
N-(2-hydroxy-2-phenylethyl)-5-(methoxymethyl)-N-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-cyclohexyl-3-[(dimethylamino)methyl]-N-(pyridin-3-ylmethyl)benzamide
5-(4-benzylpiperidin-1-yl)-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
4-(3-chloro-2-methylbenzoyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(2-methoxyphenyl)ethan-1-one
2-methoxy-3-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
N-(4-fluorophenyl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
N-{1-oxaspiro[4.5]decan-3-yl}pyrazin-2-amine
(3aS,6aS)-2-(5-chloro-2-fluorobenzoyl)-5-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]propan-1-one
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperazine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-5-ethyl-1,3,4-oxadiazol-2-amine
4-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3-dimethylpiperazin-2-one
5-chloro-N-methyl-2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)benzamide
2-(cyclopropylmethyl)-N-[2-(dimethylamino)ethyl]-N,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-[(3R,4S)-1-[1-(3,4-difluorophenyl)piperidin-4-yl]-4-(dimethylamino)piperidin-3-yl]propanoic acid
2-(azocan-1-yl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)acetamide
4-cyclopentyl-N-[2-(pyrazin-2-yl)ethyl]pyrimidin-2-amine
4-{[3-(trifluoromethyl)phenyl]methyl}-1-[(2,3,6-trifluorophenyl)methyl]-1,4-diazepan-5-one
1-{2-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}azepan-2-one
1-[(3-fluorophenyl)methyl]-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-6-oxopiperidine-3-carboxamide
6-methoxy-N-[(1-methyl-3-phenyl-1H-pyrazol-5-yl)methyl]pyrimidin-4-amine
methyl 3-{[5-(hydroxymethyl)furan-2-yl]methyl}-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}phenol
2,3-dimethoxy-N-propyl-N-(pyridin-3-ylmethyl)benzamide
(2R,3R)-3-(morpholin-4-yl)-1'-(pyridin-2-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[1-(1-ethyl-5-oxopyrrolidine-3-carbonyl)piperidin-4-yl]benzonitrile
N-(4-methoxy-2-methylphenyl)-3-[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]propanamide
1-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one
4-(5-ethyl-4-phenyl-1H-imidazol-2-yl)-1-(2-methylpropyl)pyrrolidin-2-one
4-(2-{3-[3-(4,6-dimethylpyrimidin-2-yl)phenyl]-1H-pyrazol-1-yl}ethyl)morpholine