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1-(2,3-dihydro-1H-inden-2-yl)-4-(3-propyl-1H-pyrazole-5-carbonyl)-1,4-diazepane
1-{3-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidine-1-carbonyl]phenyl}pyrrolidin-2-one
4-amino-N-butyl-N-[(2-methylphenyl)methyl]pyridine-2-carboxamide
N-(2-methoxyethyl)-6-methyl-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
3-methyl-6-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}pyridazine
2-ethyl-4-methyl-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-1,3-oxazole-5-carboxamide
N-benzyl-2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]acetamide
2-ethyl-N-[(2-fluorophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-(5-benzyl-1,3,4-thiadiazol-2-yl)-2-methyl-5-oxo-1,4-diazepane-1-carboxamide
1-{2-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)ethyl]piperidin-1-yl}-2-methylpropan-1-one
2-(3-chloro-4-ethoxyphenyl)-1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazole
2-methoxy-N-{2-methyl-3-[({2-[(3-methylpyridin-4-yl)amino]ethyl}carbamoyl)amino]phenyl}acetamide
1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-(1-methylpyrrolidin-3-yl)piperidine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-7-(3-methoxypropanamido)-1-methyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
2-[4-(pyrrolidin-3-yl)piperidin-1-yl]pyrimidine
2-methoxyethyl (3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carboxylate
2-({[(1R,2R)-2-hydroxycyclohexyl]methyl}amino)-N-[2-(2-methoxyphenyl)ethyl]acetamide
4-acetyl-N-[3-methyl-1-(2-methylphenyl)-1H-pyrazol-5-yl]-1,4-diazepane-1-carboxamide
6-{3-[1-(dimethylamino)ethyl]phenyl}-N2,N2-dimethylpyrimidine-2,4-diamine
1,5-dimethyl-4-({2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
5-(piperidin-1-yl)-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
3-(1-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-3,4-dihydroquinazolin-4-one
1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]-2-(1-methyl-1H-indol-3-yl)ethan-1-one
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
2-(dimethylamino)-N-[3-(4-methylbenzenesulfonamido)propyl]-2-(2-methylphenyl)acetamide
2-cyclopentyl-N-({5-[(oxolan-2-ylmethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)acetamide
1-(1-{[5-(4-chlorophenyl)furan-2-yl]methyl}piperidin-3-yl)-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
methyl (2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-{[2-(6-methylpyridin-2-yl)ethyl]carbamoyl}pyrrolidine-2-carboxylate
5-methyl-N-[(3R,4S)-1-[2-(2-oxopyrrolidin-1-yl)ethyl]-4-(propan-2-yl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
N-[(2,6-dimethoxyphenyl)methyl]-5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[(5-methylfuran-2-yl)methyl]benzamide
4-{2-[3,5-bis(trifluoromethyl)phenyl]acetyl}piperazine-2-carboxylic acid
(1-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}piperidin-4-yl)methanol
5-ethyl-1'-(3-fluoro-4-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(1H-pyrazol-3-yl)-N-{3-[(trifluoromethyl)sulfanyl]phenyl}piperidine-1-carboxamide
1-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-3-amine
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-6-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-{2-[(3,6-dimethylpyrazin-2-yl)amino]ethyl}pyridine-3-carboxamide
[(4aS,8aR)-6-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]-decahydro-1,6-naphthyridin-4a-yl]methanol
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-1H-pyrazole-4-carbonyl)-4-(propan-2-yl)piperazine
2-({4-[6-(methoxymethyl)pyrimidin-4-yl]piperazin-1-yl}methyl)benzonitrile
{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}[1-(1H-imidazol-1-yl)propan-2-yl]amine
N-[2-(4-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
3-[(2-methyl-1,3-benzoxazol-5-yl)methyl]-1λ6-thiane-1,1-dione
(2S,4S)-1-cyclopentyl-N-ethyl-4-{2-[methyl(phenyl)amino]acetamido}pyrrolidine-2-carboxamide
N-[2-(dimethylamino)-1-phenylethyl]-N-methyl-4-(4H-1,2,4-triazol-4-yl)benzamide
1-(2-methylpyridin-4-yl)-4-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}-1,4-diazepane
1-{2-chloro-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-N-(4-fluorophenyl)piperidin-3-amine
5-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazole-4-carboxamide