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dimethyl[2-({[4-(pyrimidin-5-yl)phenyl]methyl}(thiophen-3-ylmethyl)amino)ethyl]amine
(3R,4S)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(4-methoxyphenyl)pyrrolidin-3-amine
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N,1-dimethyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)pyrrolidine-3-carboxamide
2-butyl-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-acetyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]benzamide
3-fluoro-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-(3-methylphenoxy)piperidine-4-carboxylic acid
N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
3-[({5-methyl-1-[2-(piperidin-1-yl)ethyl]-1H-pyrazol-4-yl}methyl)amino]-1λ6-thiolane-1,1-dione
4-(2-methoxyphenoxy)-1-[2-(methylsulfanyl)benzoyl]piperidine
N-[(3S,5S)-1-acetyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1-phenyl-1H-pyrazole-4-carboxamide
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-(thiophene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperazin-1-yl}-2-[(3-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
6-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(oxolan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-[2-(dimethylamino)ethyl]-N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)piperazine-1-carboxamide
5-(3-methoxyphenyl)-4-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-2-(pyridin-4-yl)pyrimidine
(4aR,7aS)-4-(2-hydroxybenzoyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-6-(piperidin-1-yl)pyrimidin-4-amine
methyl (2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-{[(3-methylpyridin-2-yl)methyl]carbamoyl}pyrrolidine-2-carboxylate
N,8-dimethyl-3-[(5-oxo-1,4-diazepan-1-yl)methyl]-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-(4-aminopyrimidin-2-yl)-4-[(4-chlorophenyl)methyl]piperidine-4-carboxylic acid
{4-[2-(4-fluorophenyl)piperidine-1-carbonyl]phenyl}methanol
(2R)-2-phenyl-2-{[7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}ethan-1-ol
N-methyl-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}thian-4-amine
5-chloro-2-methoxy-N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
5-[(2E)-but-2-en-1-yl]-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazole-2-carboxamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-propylacetamide
2-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4,6-bis(propan-2-yl)phenol
1-(3,5-dimethylphenyl)-4-[4-(pyrrolidin-3-yl)benzoyl]piperazin-2-one
N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2,3-dihydro-1-benzofuran-7-carboxamide
[(2S,4R)-4-(dimethylamino)-1-[(2E)-2-methylpent-2-en-1-yl]pyrrolidin-2-yl]methanol
6-(4-benzylpiperidine-1-carbonyl)-5-methyl-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidin-4-amine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(4-phenylpiperidin-1-yl)acetamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-[(4-methylphenyl)methyl]-5-oxopyrrolidine-3-carboxamide
2-{[4-(1,3-dimethyl-1H-pyrazol-5-yl)-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-(6-chloro-2-methylpyridin-3-yl)-3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]urea
N,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[(1-methylpiperidin-4-yl)methyl]quinoline-4-carboxamide
3-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-N,N-dimethylpropane-1-sulfonamide
1-{3-[(cycloheptylamino)methyl]phenoxy}-3-(4-ethylpiperazin-1-yl)propan-2-ol
5-cyclopropyl-3-({5-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-4-phenyl-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazole
9-methoxy-4-(1H-pyrrol-2-ylmethyl)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-({1-[4-(methylsulfanyl)butan-2-yl]piperidin-4-yl}oxy)-N-(pyridin-4-ylmethyl)benzamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidine
5-cyclopropyl-N-[2-(diethylamino)ethyl]-N-methyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
5-methyl-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-1,2-oxazole-3-carboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(1H-imidazol-1-yl)acetamide
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]azetidine-2-carboxylic acid
4-[4-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)piperazin-1-yl]quinazoline