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(3S)-N,N-dimethyl-1-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}azepan-3-amine
1-[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(pyridin-3-yl)propan-1-one
4-benzyl-3-ethyl-1-[4-(hydroxymethyl)benzoyl]-1,4-diazepan-5-one
N,N-dimethyl-5-{[(1R,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyrimidin-2-amine
N-[(3S,4R)-1-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-4-propylpyrrolidin-3-yl]acetamide
3-({4-[3-(4-ethyl-4-methylpiperidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
1-(2-fluorophenyl)-N-[2-(2-hydroxyethoxy)ethyl]-2,2-dimethylcyclopropane-1-carboxamide
2-(2-aminoethyl)-N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}quinazolin-4-amine
(3S,4R)-4-(3-fluorophenyl)-1-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
N-[5-carbamoyl-2-(2-methylpiperidin-1-yl)phenyl]-3-hydroxypyridine-2-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
1-(cyclohexylmethyl)-N-(diphenylmethyl)-6-oxopiperidine-3-carboxamide
8-cyclopropanecarbonyl-2-(4-methylpyrimidine-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(2-benzyl-1,3-thiazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
(2E)-N-{[7-(5-acetylthiophene-3-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-phenylprop-2-enamide
9-(oxan-2-ylmethoxy)-4-[4-(1H-pyrazol-1-yl)benzoyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(1R,2S)-2-(methoxymethyl)cyclopentyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-{[4-(5-chlorothiophen-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
N-[(3-propyl-1,2-oxazol-5-yl)methyl]-6-(pyrrolidin-1-yl)pyridine-3-carboxamide
3-[1-(1-ethyl-2-oxo-1,2-dihydropyridin-4-yl)-N-(2-phenylethyl)formamido]propanamide
(1R,5R)-6-{imidazo[1,2-a]pyridine-3-carbonyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-[2-(2-chlorophenyl)ethyl]-11-(4-propylpiperazin-1-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-cyclopentyl-N5-(diphenylmethyl)-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-({4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(4-chlorophenyl)-4-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}morpholine
1-{1-[6-(4,4-dimethylpiperidin-1-yl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]-N-[2-(6-methylpyridin-2-yl)ethyl]piperidin-4-amine
3-({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)-2,2-dimethylpropan-1-ol
2-cyclopentyl-1-[7-(6,7-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
2-[(cyclopropylmethyl)sulfanyl]-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}ethan-1-one
methyl 4-{[(3aS,6aR)-3-cyclopentyl-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]methyl}benzoate
5-ethyl-2,3-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(3-fluoropyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]azetidin-3-ol
5-chloro-3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
2-methyl-7-(2,5,7-trimethylquinoline-4-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-chloro-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-2-methylbenzamide
N-(5-{3-[1-(dimethylamino)ethyl]phenyl}pyridin-2-yl)cyclopropanecarboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)acetamide
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl)(1,3-thiazol-4-ylmethyl)amine
1-[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-{[8-(3,4-dimethylbenzoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}pyridine-2-carboxamide
2-{3-[(2-fluorophenyl)methyl]-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl}acetic acid
N'-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]ethanediamide
N-[2-(3-fluorophenyl)ethyl]-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
N-[1-(6-methoxynaphthalen-2-yl)ethyl]-2-(piperidin-4-yl)acetamide
1-[3-(methylsulfanyl)propyl]-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pent-4-en-1-one