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1-(2-methoxy-5-{[methyl(2-methylpropyl)amino]methyl}phenoxy)-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
1-(3-chlorophenyl)-4-({4-[(1-cyclohexanecarbonylpiperidin-4-yl)oxy]phenyl}methyl)piperazine
(3S,4R)-4-(2-methoxyphenyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidine-3-carboxylic acid
N-cyclopropyl-1-[1-(3-methoxypyridine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
4-[1-({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)ethyl]hepta-1,6-dien-4-ol
N-[1-ethyl-2-(2-fluorophenyl)-7-(morpholine-4-carbonyl)-1H-1,3-benzodiazol-5-yl]acetamide
1-cyclopropyl-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methyl-6-oxopiperidine-3-carboxamide
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-5-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[3-(methoxymethyl)phenyl]-2-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}acetic acid
4-{[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}pyrrolidin-2-one
4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-5-methyl-3-phenyl-1,2-oxazole
1-[3-({[(3-fluorophenyl)methyl]amino}methyl)-7-methylquinolin-2-yl]piperidin-4-ol
(4aS,7aR)-1-[(3,5-dimethylphenyl)methyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,4R)-3-cyclopropyl-1-(4-ethyl-5-methylthiophene-3-carbonyl)-4-methylpyrrolidin-3-ol
1-(2-{[(6-methylpyrimidin-4-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
4-[4-(benzyloxy)-3-fluorophenyl]-6-(methoxymethyl)pyrimidine
2-{4-[(3,5-difluorophenyl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(3S,4R)-3-cyclopropyl-4-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetamido}-N,N-dimethylpyrrolidine-1-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[1-methyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
3-amino-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
2-(1-tert-butyl-1H-pyrrole-3-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2,3-dimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]quinoxaline-6-carboxamide
N-[3-(azepane-1-carbonyl)phenyl]-3-methoxypiperidine-1-carboxamide
4-[1-(furan-2-ylmethyl)piperidin-4-yl]-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-[2-(butan-2-yl)phenoxy]ethan-1-one
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethan-1-one
1-[1-(2-phenylethyl)-5-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,4-diazepan-5-one
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-4-methoxybenzamide
6-oxo-1-(prop-2-en-1-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]piperidine-3-carboxamide
N-({5-[(2-chloro-6-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
1-(4-acetyl-4-phenylpiperidin-1-yl)-4-(1H-imidazol-1-yl)butan-1-one
2-(1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,3-benzothiazole
N-cyclopropyl-1-(2-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
N-({3-[1-(cyclohex-2-en-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]-1,2-oxazol-5-yl}methyl)-N-methylacetamide
1-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(2-phenoxyethyl)piperazine
2-[2-(benzyloxy)ethyl]-8-methyl-2,8-diazaspiro[4.5]decane
2-(2-oxopyrrolidin-1-yl)-N-{[1-(phenoxymethyl)cyclopropyl]methyl}propanamide
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(5-propylpyrimidin-4-yl)piperidin-4-amine
(4S)-4-hydroxy-3,3,4-trimethyl-N-[2-(thiophen-2-yl)ethyl]piperidine-1-carboxamide
2-amino-4-[3-(2-hydroxyethoxy)phenyl]-6-(2-methylphenyl)pyridine-3-carbonitrile
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
[(5-ethylpyridin-2-yl)methyl](2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amine
N-[3-(benzylsulfanyl)propyl]-2-(2-oxopiperidin-1-yl)acetamide
(3aR,6aS)-5-(1H-1,3-benzodiazol-2-ylmethyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2R,3R,6R)-5-[1-(methoxymethyl)cyclobutanecarbonyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[4-(2-fluorophenoxy)phenyl]-1-(furan-3-carbonyl)piperidine-4-carboxamide
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-1-ethyl-N-(2-hydroxyethyl)-1H-pyrazole-4-carboxamide
3-(piperidin-4-ylmethyl)-N-[(2-propyl-1,3-thiazol-4-yl)methyl]benzamide