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N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-N'-(4-methylphenyl)propanediamide
5-({[(3-{2-[4-(2,6-dimethoxybenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
4-{2-[benzyl(methyl)carbamoyl]ethyl}-N-(2-phenylethyl)piperidine-1-carboxamide
N-[1-(4-chlorophenyl)-5-oxopyrrolidin-3-yl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
4-[(4-fluorophenyl)methyl]-1-[2-(2-oxopyrrolidin-1-yl)ethyl]-3-(propan-2-yl)-1,4-diazepan-5-one
(2S)-2-[(1-cyclopropanecarbonylpiperidin-4-yl)formamido]-3-(4-hydroxyphenyl)propanoic acid
1-{2-oxo-2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}piperidin-2-one
3-[({[1-(ethoxymethyl)cyclopropyl]methyl}carbamoyl)methyl]-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
2-({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)acetamide
N,N-diethyl-1-[1-(quinolin-4-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
1-[2-(1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
4-{1-[(3S,4R)-4-ethoxyoxolan-3-yl]-4-phenyl-1H-imidazol-5-yl}-2-(propan-2-yl)pyrimidine
N-({7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-1-methylpiperidine-3-carboxamide
(2-ethoxy-5-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}phenyl)methanol
4-methyl-3-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)benzene-1-sulfonamide
9-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
(1S,5R)-3-(1-methyl-1H-pyrazole-4-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carboxamide
4-{[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
ethyl 4-[3-(carbamoylmethyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]piperidine-1-carboxylate
1-(2-{[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-5-yl]formamido}ethyl)piperidine-3-carboxamide
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-benzofuran-3-carboxamide
N-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}propanamide
N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
5-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-3-[3-(dimethylamino)propyl]-5-[(3-fluorophenyl)methyl]imidazolidine-2,4-dione
N-[(2-chloro-4-fluorophenyl)methyl]-2-[methyl(piperidin-4-yl)amino]acetamide
5-(naphthalen-1-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-(1-methoxypropan-2-yl)-1-[4-(3-methylphenyl)phenyl]piperidin-4-amine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-(2-methylphenyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
methyl 3-(4-fluorobenzoyl)-9-[2-(morpholin-4-yl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-[6-(piperidine-1-carbonyl)pyrazin-2-yl]thiophene-2-carboxylic acid
3-{2-[2-(3-chloro-4-hydroxyphenyl)-1H-imidazol-1-yl]phenyl}-N,N-dimethylpropanamide
3-{1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1,3-oxazolidin-2-one
1-tert-butyl-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
1-[3-(cyclohexylsulfanyl)propyl]-3-(2-hydroxypyridin-3-yl)urea
N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
4-{4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-3,5-dimethyl-1H-pyrazole
6-[4-(morpholine-4-carbonyl)piperidine-1-carbonyl]pyridin-2-amine
4-(1-methyl-1H-imidazol-2-yl)-1-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1H-1,2,3-triazole
2-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
4-(2,3-dihydro-1H-isoindol-2-yl)-N-[(1-methylpyrrolidin-3-yl)methyl]butanamide
1-acetyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidine-3-carboxamide
1-[(1S,5R)-6-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4-(2-methylpyridin-4-yl)-1,4-diazepane
4-(4-fluorophenyl)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-4-ol
1-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butan-1-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2,4-difluoro-3-methoxybenzoyl)piperidin-3-ol
1-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide