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N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1-phenyl-1H-1,2,3-triazole-4-carboxamide
2-[1-(dimethyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]-5-fluoro-1H-1,3-benzodiazole
2-{4-[4-(morpholin-4-yl)phenyl]-1H-pyrazol-1-yl}-N-[1-(propan-2-yl)-1H-pyrazol-5-yl]acetamide
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[2-(trifluoromethyl)morpholin-4-yl]propan-1-one
2-hydroxy-1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-4-methylpentan-1-one
1-[1-(4-methylpiperazine-1-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
2-({5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propan-1-ol
4-[(3,5-dichloropyridin-4-yl)methyl]-N-(4-fluorophenyl)piperazine-2-carboxamide
1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-2-(3-methoxyphenyl)azetidine
N-{2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}acetamide
3-chloro-6-{4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}pyridazine
4,6-dimethyl-3-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-1,2-dihydropyridin-2-one
3-{4-phenyl-1-[3-(pyridin-3-yl)propyl]-1H-imidazol-5-yl}pyridine
2-[4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperazin-1-yl]pyrimidine
1-[(3-fluorophenyl)methyl]-4-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperazine
N,N-dimethyl-5-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}pyridin-2-amine
4-[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]-N-[2-(4-methoxyphenyl)ethyl]piperidine-1-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(3-fluorophenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
2-{4-[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyrimidin-5-yl}acetic acid
2-[(2-ethylpyrimidin-5-yl)methyl]-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
2-[4-(3,4-difluorophenyl)-1H-pyrazol-1-yl]-N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
N-[3-(2-chlorophenoxy)propyl]-N-methyl-2-propyl-1,3-thiazole-4-carboxamide
9-hydroxy-3-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
5-[2-(cyclopropylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(4aS,8aS)-4a-hydroxy-7-(5-methoxyfuran-2-carbonyl)-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
N-[2-(3-benzyl-1H-1,2,4-triazol-5-yl)phenyl]-N-methylthiophene-2-carboxamide
2-ethoxy-1-{4-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]piperidin-1-yl}ethan-1-one
3-{2-[(pyridin-3-yl)amino]ethyl}-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
ethyl[(4-methyl-1H-imidazol-2-yl)methyl]({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amine
2-{3-[(2-methoxyphenyl)methoxy]phenyl}-N-methylpyridine-3-carboxamide
N-{[7-(2-methoxy-2-phenylacetyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-2-yl)piperidin-4-ol
1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(1H-1,2,3,4-tetrazol-5-yl)piperidine
N-ethyl-N-methyl-1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-sulfonamide
1-{3-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]phenyl}ethan-1-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
3-({2-[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
[(1-methyl-1H-imidazol-2-yl)methyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)(propan-2-yl)amine
3-[(3R,4S)-4-(dimethylamino)-1-(2-methoxy-4-methylbenzoyl)piperidin-3-yl]propan-1-ol
7,7-dimethyl-2-{2-[(pyridin-3-yl)amino]ethyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(1S,5R)-3-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
9-[2-(2-oxopyrrolidin-1-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-1-(2-methoxyethyl)pyrrolidin-2-one
N-[(3R,4S)-4-cyclopropyl-1-[(2-fluoro-4-methoxyphenyl)methyl]pyrrolidin-3-yl]acetamide
6-methyl-4-(4-methyl-1H-imidazol-5-yl)-N-[2-(3-methylthiophen-2-yl)ethyl]-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(2R,6R)-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
ethyl 4-[(2-chlorophenyl)methyl]-1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]piperidine-4-carboxylate
5-[1-(2,5-difluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-2-ethylpyrimidine