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5-{2-[4-(cyclopropylmethyl)piperazin-1-yl]pyrimidin-4-yl}-2-ethoxybenzoic acid
N-[1-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2H-1,3-benzodioxole-5-carboxamide
2-(3-methylthiophen-2-yl)-1-{1-oxaspiro[4.4]nonan-3-yl}-1H-imidazole
1-{1'-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-(1-{1-[3-(2-methoxyphenyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
N-methyl-2-(methylsulfanyl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrimidine-5-carboxamide
4-{2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]acetyl}-1,4-diazepane-1-carbaldehyde
3-{1-[(2S)-2-amino-3-(1H-imidazol-4-yl)propanoyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
8-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
3-cyano-5-fluoro-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]benzamide
4-[(2-methylprop-2-en-1-yl)oxy]-N-[2-(morpholin-4-yl)butyl]benzamide
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-(3-methoxyphenyl)-N-methylpropanamide
2-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]pyrimidin-4-amine
N-ethyl-1-propyl-N-(pyridin-4-ylmethyl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(2,5-dimethoxybenzoyl)piperidine-3-carboxylate
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-methoxypyridine-2-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
N-cyclopropyl-5-(6-methyl-2-propylpyrimidin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-[(1S,5R)-6-benzyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4,6-dimethylpyridine-3-carbonitrile
3-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]urea
4-{[(2-methoxyphenyl)methyl]amino}-5-methyl-N-(oxolan-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
{1-[1-(methylsulfanyl)propan-2-yl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
8-(2,3-dihydro-1-benzothiophene-2-carbonyl)-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-methoxyethyl)-4-(4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}piperidin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
(1s,4s)-N1-{1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}cyclohexane-1,4-diamine
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
(2S,4S)-4-amino-1-{[5-(3-chloro-4-methylphenyl)furan-2-yl]methyl}pyrrolidine-2-carboxylic acid
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(4-methylpiperidin-1-yl)acetamide
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2,3-difluorophenyl)ethan-1-one
2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidine
N-methyl-N-[3-(oxolan-2-yl)propyl]-2-(trifluoromethyl)pyrimidin-4-amine
4-[(2,4-dimethyl-1H-imidazol-1-yl)methyl]-5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazole
1-(1,3-benzothiazol-2-ylmethyl)-1-methyl-3-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]urea
ethyl 5-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2-(N-methylmethanesulfonamido)ethyl]propanamide
N,N-dimethyl-1-(5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carbonyl)pyrrolidin-3-amine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N3-(cyclohexylmethyl)-1-cyclopropyl-N5-[(1R)-1-(3-methoxyphenyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-{[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl](methyl)amino}-N-methylbutanamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
N,N-dimethyl-5-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-1,3-thiazol-2-amine
5-(1H-imidazol-2-yl)-2-(3-methoxyphenyl)-1,3-thiazole
5-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(pyridin-4-ylmethyl)amino]methyl}piperidin-2-one
3-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-4-methoxybenzene-1-sulfonamide
methyl 4-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}methyl)thiophene-2-carboxylate
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
4-[butyl(pyridin-3-ylmethyl)carbamoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylic acid
1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine