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N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-3-one
4-[2-(2-aminoethyl)quinazolin-4-yl]-1λ6-thiomorpholine-1,1-dione
5-[(4-chloro-1H-pyrazol-1-yl)methyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-(dimethyl-1,3-thiazol-4-yl)-N-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]acetamide
N-[(1S,2R)-2-[(2,3-dihydro-1H-inden-2-yl)amino]cyclobutyl]pyridine-3-sulfonamide
N-(5-{[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}thiophen-2-yl)acetamide
3-(4-chloro-1H-pyrazol-1-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)propanamide
(3S,4R)-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
(3S,4R)-1-{[(cyclohexylmethyl)carbamoyl]methyl}-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
methyl 6-[(4-methoxy-2,3-dimethylphenyl)methyl]-2-[(propan-2-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N,N-dimethyl-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]azepan-4-amine
1-{[4-(4-chlorophenoxy)phenyl]methyl}-3-[(dimethylamino)methyl]piperidin-3-ol
6-methyl-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
3-(8-methoxy-2-methylquinolin-5-yl)-1-methyl-6-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-(cyclohexyloxy)-3-({8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}amino)propan-2-ol
1-[(3-fluorophenyl)methyl]-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazine
methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl){[4-(2-methylphenyl)phenyl]methyl}amine
3-methyl-8-[4-(1H-pyrazol-4-yl)butanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}sulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(2,5-dioxoimidazolidin-4-yl)acetamide
2-{4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)-6-azaspiro[2.5]octane-1-carboxamide
5-fluoro-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-(pyrrolidin-1-yl)pyrimidin-2-amine
1-[2-(4-methoxyphenyl)ethyl]-N-[(5-methylfuran-2-yl)methyl]-5-(4-methylpiperidine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
methyl 5-[(2-hydroxy-7-methylquinolin-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
5-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridine-2,4-diol
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
8-[1-(3-chlorophenyl)piperidin-4-yl]-2,8-diazaspiro[4.5]decan-3-one
3-{2,7-diazaspiro[4.5]decan-2-yl}-N-(3,5-dimethylphenyl)-3-oxopropanamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-(3-fluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(3-phenylpropyl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)morpholine-2-carboxamide
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]propan-1-one
1-(cyclopropylmethyl)-4-[2-(5-methyl-1H-pyrazol-1-yl)ethyl]-2-(propan-2-yl)-1,4-diazepane
N-(3-hydroxy-3-phenylpropyl)-N-methyl-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
1-(1-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-phenylpiperidin-4-yl)ethan-1-one
ethyl 3-benzyl-1-(pyridin-2-ylmethyl)piperidine-3-carboxylate
6-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-3-(8-methoxy-2-methylquinolin-5-yl)-1-methyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-methyl-N-(4-{2-[3-(pyridine-2-carbonyl)piperidin-1-yl]acetamido}phenyl)acetamide
1-phenyl-2-(7-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethane-1,2-dione
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-(1H-pyrazol-1-yl)benzamide
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)morpholine
N-benzyl-N,1-dimethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-methyl-1-[2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidine-3-carboxamide
5-fluoro-2-{3-[2-(pyridin-4-yl)-1H-imidazol-1-yl]propyl}-1H-1,3-benzodiazole
8-[2-(methylamino)pyridine-4-carbonyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-cyclopentyl-N3-methyl-N5-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
N-[1-(2,5-dimethylphenyl)ethyl]-5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide