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(2S)-3-hydroxy-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(methylamino)propan-1-one
(2S,4S)-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}-N-methyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-[2-(methylsulfanyl)benzoyl]piperidine
2-(4-fluorophenyl)-4-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]morpholine
1-[5-({[2-(1H-imidazol-1-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(piperidin-1-yl)propan-2-ol
1-({[(4,6-dimethylpyridin-2-yl)methyl](methyl)carbamoyl}methyl)piperidine-4-carboxamide
(4aR,7aS)-1-ethyl-4-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-phenylethyl)-1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
(4aR,8aR)-2-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1-methylimidazolidin-2-one
4-[5-(methoxymethyl)thiophene-2-carbonyl]-7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
2-methyl-4-{3-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]phenyl}but-3-yn-2-ol
1-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-3-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}urea
N'-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-N,N-dimethylbutanediamide
2-ethyl-5-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
4-cyclohexyl-N-[4-(2-oxopyrrolidin-1-yl)phenyl]piperazine-1-carboxamide
(8R,9aS)-2-[2-(2-chlorophenyl)ethyl]-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
N-(1-phenylethyl)-4-(4-{[2-(piperidin-1-yl)ethyl]amino}piperidin-1-yl)benzamide
2-{[2-(dimethylamino)-4-oxo-1,3,8-triazaspiro[4.5]dec-1-en-8-yl]methyl}benzonitrile
(4aS,8aR)-6-[4-(aminomethyl)benzoyl]-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
3-{[(adamantan-1-yl)amino]methyl}-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
3-({[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
7-[2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-ethyl-4-[4-(4-fluorophenoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
7-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
(3S,4S)-1-(2-{[(3-chlorophenyl)methyl]carbamoyl}ethyl)-4-propylpyrrolidine-3-carboxylic acid
1-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
5-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-(2-chlorophenoxymethyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-cyclohexyl-5-{[3-(pyrimidin-4-yl)piperidin-1-yl]methyl}pyrimidine
7-(2-phenylpyrrolidine-1-carbonyl)-1,3-diazepane-2,4-dione
[(2S,6S)-4-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-hydroxypropan-1-one
1-methyl-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-butyl-2-[methyl({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl})amino]acetamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-(2-methoxyethyl)-N-methyl-1,3-oxazole-4-carboxamide
1-[1-ethyl-5-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
3-chloro-2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-{2-[2-(dimethylamino)ethyl]morpholin-4-yl}-3-(4-methylphenyl)propan-1-one
2-benzyl-N-[2-(methylsulfanyl)ethyl]-1,3-benzoxazole-5-carboxamide
N-(1-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-2-carboxamide
2-{8-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1-ethyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
1-{[4-(methylsulfanyl)phenyl]methyl}-4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
1-{2-[ethyl(methyl)amino]acetyl}-4-(2-fluoro-5-methylphenoxy)piperidine-4-carboxylic acid
1-[1-(1-carbamoylcyclopropanecarbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
3-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}-N,N-dimethylpiperidine-1-carboxamide
2-methoxy-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide