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1-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-N-(3-methylbutan-2-yl)piperidin-4-amine
2-(benzyloxy)-N-(isoquinolin-5-ylmethyl)-N-methylacetamide
7-fluoro-N-[(5-methylpyrazin-2-yl)methyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(3R,4R)-1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
5-propyl-N-[2-(pyrazin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
methyl 4-(4-{[3-(2-ethoxy-2-oxoethyl)morpholin-4-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
4-({[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]amino}methyl)-2-methoxyphenol
3-[(3R,4S)-1-[(2,4-dimethylphenyl)carbamoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
12-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-15-methyl-9-(pyridin-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
7-(4-methoxybenzoyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(4-chloro-1H-pyrazol-1-yl)-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}propan-1-one
1-{4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-2,2-diphenylethan-1-ol
3-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{[2-(methylsulfanyl)phenyl]methyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
1-amino-N-{[1-(2,3-dihydro-1H-inden-2-yl)pyrrolidin-3-yl]methyl}cyclopentane-1-carboxamide
N-(2-methoxyphenyl)-2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-carboxamide
2-(butylsulfanyl)-6-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyrimidin-4-amine
N-(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}pyrimidin-2-yl)benzenesulfonamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-2-(1,3-thiazol-2-yl)pyrrolidine-1-carboxamide
2-methyl-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-6-(piperidin-4-yl)pyrimidin-4-amine
(4-{[1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-2-methoxypyridine
N-ethyl-3-({[1-(3-fluoro-4-methoxyphenyl)ethyl]carbamoyl}amino)-2-methylbenzamide
1-tert-butyl-N-{1-[(4-chlorophenyl)methyl]cyclopropyl}-5-oxopyrrolidine-3-carboxamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(2,5-dioxoimidazolidin-4-yl)acetamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
ethyl 5-(2,6-dimethylpyrimidine-4-carbonyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
5-[1-(3-chlorobenzoyl)pyrrolidin-2-yl]-N,N-diethylthiophene-2-carboxamide
{2-ethoxy-5-[1-(1,2-oxazol-3-ylmethyl)-4-phenyl-1H-imidazol-5-yl]phenyl}methanol
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N-propylpiperidine-1-carboxamide
5,6-dimethyl-3-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-(1-cyclohexyl-5-{[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]methyl}-1H-1,2,4-triazol-3-yl)acetamide
1,6-dimethyl-4-oxo-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1,4-dihydroquinoline-3-carboxamide
1-(oxan-4-yl)-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperazine
1-(4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)-4-phenylpiperidine-4-carbonitrile
6-[(2-ethyl-1,3-thiazol-4-yl)methyl]-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
N-[2-(4-chlorophenoxy)ethyl]-N-(furan-2-ylmethyl)oxane-4-carboxamide
N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
4-[1-(3-methylpyridin-4-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]-1,2-dihydroquinolin-2-one
3-(furan-2-yl)-4-[4-(1H-1,2,4-triazol-1-yl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-methyl-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}urea
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-[(5-fluoro-2-methylphenyl)methyl]-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,3,4-trimethoxybenzamide
(8aS)-2-[3-oxo-3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-cyclopentyl-5-methyl-4-[(thiophen-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide