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N-[(4-fluorophenyl)methyl]-N,7-dimethylimidazo[1,2-a]pyridine-2-carboxamide
ethyl 3-({1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)butanoate
4-[5-(2-chlorophenyl)-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl]-1-methylpyrrolidin-2-one
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-imidazol-4-yl)ethyl]amine
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(oxan-4-ylmethyl)acetamide
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,2-oxazole-3-carboxamide
[(3S,5R)-5-[(dimethylamino)methyl]-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]methanol
N,N-dimethyl-3-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]aniline
{2-[4-(2-chlorophenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}urea
N-[3-(4-fluorophenyl)phenyl]-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine-3-carboxamide
(1,3-benzothiazol-2-ylmethyl)({[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
(2S)-2-[2-(2-chlorophenyl)-1H-imidazol-1-yl]-4-methylpentan-1-ol
N-[3-(3-methoxyphenyl)phenyl]-1-propylpiperidine-4-carboxamide
N-(4-fluoro-2-methylphenyl)-2-[2-(pyridin-3-yloxy)acetamido]propanamide
2-(3-chloro-2-fluorophenyl)-1-methyl-1H-imidazole
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(hydroxymethyl)-N-(2-methoxyethyl)-1H-1,3-benzodiazole-5-carboxamide
7-cyclopentyl-2-(6-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2,3,5-trimethyl-N-[3-(4H-1,2,4-triazol-4-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
methyl 1-(2-methoxyethyl)-3-(3-methylbutanamido)-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(butylsulfanyl)-5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}pyrimidine
8-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[(3,4-dimethoxyphenyl)methyl]-N-methyl-2-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}quinazolin-4-amine
4-({[5-(naphthalen-1-yl)-1,2,4-triazin-3-yl]amino}methyl)-1,2-dihydrophthalazin-1-one
1-methyl-3-[2-(morpholin-4-yl)-2-oxoethyl]-3-(4-phenylphenyl)pyrrolidine-2,5-dione
3-[(3-hydroxypiperidin-1-yl)sulfonyl]-N-(oxan-4-yl)benzamide
5-cyclohexaneamido-1-(2-methoxyethyl)-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1H-1,3-benzodiazole-7-carboxamide
8-methoxy-N-[(5-methylpyrazin-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-{3-[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]propyl}-3,5-dimethyl-1,2-oxazole
1,3-dimethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-cyclopentyl-N-ethyl-4-oxo-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridine-3-carboxamide
3-(1-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)pyridine
1-cyclopentyl-N3-ethyl-4-oxo-N5-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-3-(pyridin-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(2-fluorophenyl)-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}cyclopropane-1-carboxamide
5-[4-(diphenylmethyl)piperazine-1-carbonyl]-4-methylpyrimidine
{[4-({1-[(5-chlorothiophen-2-yl)sulfonyl]piperidin-4-yl}oxy)phenyl]methyl}(methyl)(quinolin-6-ylmethyl)amine
(3S,4S)-1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-fluoro-1,3-benzothiazol-2-amine
8-(2-amino-2-methylpropyl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-({5-[1-(3-chlorophenyl)-1H-pyrazol-4-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
4-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-4-oxobutane-1-sulfonamide
3-cyclopentyl-1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
N-{[1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
2-methyl-8-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-butyl-3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-3-ylmethyl)propanamide
(1R,4S)-2-{2-[3-(trifluoromethyl)phenyl]pyridine-3-carbonyl}-2-azabicyclo[2.2.1]heptane
methyl (2S,4R)-1-[(3-chloro-4,5-diethoxyphenyl)methyl]-4-hydroxypyrrolidine-2-carboxylate