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{4-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
3-methyl-1-(1-{6-[methyl(pyridin-3-ylmethyl)amino]pyridine-3-carbonyl}piperidin-3-yl)butan-1-one
N-ethyl-5-[(4-{5-methylthieno[2,3-d]pyrimidin-4-yl}piperazin-1-yl)methyl]pyrimidin-2-amine
3-({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)propan-1-ol
(2R,3R,6R)-5-benzyl-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{[3-(2-aminoethyl)phenyl]methyl}-1-phenylpiperazin-2-one
5-[3-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]-1,3,4-thiadiazol-2-amine
2-(cyclopropylmethyl)-9-(4-hydroxy-3-methoxybenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-3-{[2-(3-phenylpropyl)morpholin-4-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
N-(1-cycloheptylpiperidin-3-yl)-3-acetamidopropanamide
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(oxan-3-ylmethyl)pyridin-2-amine
1,3-dimethyl-5-({[5-(naphthalen-2-yl)-1,2,4-triazin-3-yl]amino}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-{5-[1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-3-methylpiperidine-3-carboxamide
N-(1H-1,3-benzodiazol-2-yl)-2-{[(2,3-dimethylphenyl)methyl]amino}acetamide
1-(2-propoxypropanoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-(4-methoxyphenyl)-N-methyl-3-phenyl-N-(pyrimidin-4-ylmethyl)propanamide
4-(6-phenylpyridazin-3-yl)-1,4-diazepan-2-one
1-benzyl-5-(2-methyl-1,3-thiazole-4-carbonyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-amino-N-cyclopropyl-3-ethyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-4-(furan-2-ylmethyl)piperazine-1-carboxamide
3-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-3-yl]-N-(2-fluorophenyl)propanamide
1-(3,4-dimethylphenyl)-4-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-4-phenylbutane-1,4-dione
N-methyl-N-(quinolin-5-ylmethyl)-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetamide
5-cyano-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
3-[3-(2-methoxyphenoxy)propyl]-5-methyl-5-(piperidin-4-yl)imidazolidine-2,4-dione
5-butyl-4-(1-methyl-1H-pyrazole-4-carbonyl)-1-(3-phenylphenyl)piperazin-2-one
7-(2-methoxyethyl)-2-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2,7-diazaspiro[4.5]decan-6-one
1-{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}-3-(methoxymethyl)piperidine
methyl 2-(benzylsulfamoyl)-6-[(2,5-difluorophenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl 3-(2-methoxyacetamido)-1-(3-methylbutyl)-5-[(thiolan-3-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N,N-dimethyl-4-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)piperazine-1-sulfonamide
3-[1-(2,5-dimethoxyphenyl)-1H-imidazol-2-yl]-1-ethylpiperidine
(3S,4S)-1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
2-(5-methyl-1,3-oxazole-4-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-[1-(3,4-difluorophenyl)-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-6-azaspiro[2.5]octane
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-(pyridin-4-ylmethyl)-decahydro-2,7-naphthyridine-2-sulfonamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-1-methyl-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
5-(3-{1-[(2-chlorophenyl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
N-[(4-cyanophenyl)methyl]-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
5-(1-methyl-1H-imidazole-2-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
6-{imidazo[1,2-a]pyridine-3-carbonyl}-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}pyrazin-2-ol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
N,1,3-trimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
2-[(6-methoxy-2H-chromen-3-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
4-{2-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H-imidazol-1-yl}benzamide
(2S,4R)-1-(2-methylpropyl)-N-(propan-2-yl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide