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4-chloro-2-hydroxy-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]benzamide
N-{[4-(cycloheptyloxy)-3-methoxyphenyl]methyl}-N-(pyridin-2-ylmethyl)pent-4-enamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
4-ethyl-3-(piperidin-3-yl)-1-[3-(1H-pyrazol-1-yl)propyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N,5-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
N-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-2,3-dihydro-1H-inden-2-amine
1-(2,3-dihydro-1H-inden-2-yl)-4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazine
N-(furan-2-ylmethyl)-4-(1H-imidazol-1-yl)benzamide
4-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-5-methyl-2H-1,2,3-triazole
N-[2-(pyrrolidine-1-sulfonyl)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-[3-hydroxy-1-(4-methylphenyl)propyl]-N'-(4-methylphenyl)propanediamide
2-[3-(furan-2-yl)-5-(1-hydroxypropyl)-1H-1,2,4-triazol-1-yl]acetic acid
N-methyl-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidine-3-carboxamide
[(3-{2-[4-(2-chlorobenzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(thiophen-2-ylmethyl)amine
1-[(3-chlorophenyl)methyl]-4-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]piperazine
1-(4-aminopyrimidin-2-yl)-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylic acid
3-fluoro-2-methoxy-N-(2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
2-(1-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1H-1,2,3-triazol-4-yl)benzoic acid
3-(2-methylpropyl)-5-[3-(propoxymethyl)pyrrolidine-1-carbonyl]-1,2-oxazole
methyl({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})[1-(1,2-oxazol-3-yl)ethyl]amine
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]urea
8-fluoro-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}quinoline-2-carboxamide
(5S,9aS,9bS)-2-[(2-methylphenyl)methyl]-5-(thiophen-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(4-{4-[(1,3-benzothiazol-2-ylmethyl)amino]piperidin-1-yl}phenyl)-2-fluorobenzamide
N-butyl-5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
3-(thiomorpholine-4-carbonyl)-N-(2,2,2-trifluoroethyl)benzene-1-sulfonamide
N,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-(oxan-4-yl)quinoline-4-carboxamide
3-fluoro-N-(1-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
(2S)-2-amino-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-3-(1H-imidazol-4-yl)propan-1-one
4-(4-cyclopentylpyrimidin-2-yl)-2-(morpholin-4-ylmethyl)-1,4-oxazepane
3-(3-hydroxy-3-methylbutyl)-N-{1-oxaspiro[4.4]nonan-3-yl}benzamide
1-(1-methyl-5-{[methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}-1H-pyrrol-3-yl)ethan-1-one
1-(3-hydroxypropyl)-3-[2-(propan-2-ylsulfanyl)phenyl]-1-(pyridin-3-ylmethyl)urea
N,N-dimethyl-1-[2-(trifluoromethyl)benzoyl]azepan-4-amine
8-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(1-{6-[4-(dimethylamino)piperidin-1-yl]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
{1-ethyl-5-[(2-fluoro-4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
4-(dimethyl-1,2-oxazol-4-yl)-6-methyl-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,2,3,4-tetrahydropyrimidin-2-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}propan-1-one
2-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
(1S,5R)-6-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
3-[1-(6-cyanopyridin-2-yl)piperidin-3-yl]-N-(3,5-dimethoxyphenyl)propanamide
1-[4-(5-methyl-4-{[1-(thiophen-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carbonyl)piperazin-1-yl]ethan-1-one
4-(1H-1,2,3-benzotriazole-5-carbonyl)-1-(4-methoxyphenyl)-5-methylpiperazin-2-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-3-(1H-pyrazol-1-yl)propanamide
1-({5-[1-(cyclobutylmethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
N,8-dimethyl-3-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methylphenol
N-(furan-3-ylmethyl)-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide