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3-(3-fluorophenyl)-N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
(1S,5R)-3-benzoyl-6-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-5-cyclopropyl-1,3,4-oxadiazol-2-amine
2-(2-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1,2-benzothiazol-3-one
6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
[1-(2,3-dimethylquinoxaline-6-carbonyl)piperidin-4-yl](pyridin-2-yl)methanol
4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
N-({1-[(3-cyanophenyl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}methyl)thiophene-2-carboxamide
1-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[(2S)-1-methoxypropan-2-yl]urea
1-(4-chlorophenyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]cyclobutane-1-carboxamide
(2H-1,3-benzodioxol-5-ylmethyl)({4-[2-(3-methylpiperidin-1-yl)ethoxy]phenyl}methyl)amine
2-(2,3-dihydro-1,4-benzodioxin-6-yl)quinoxaline
N-[(3R,4S)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-hydroxyacetamide
11-{[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1,4,6-trimethyl-3-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-{[3-(furan-2-yl)phenyl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-methyl-5-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-3,4-dihydropyrimidin-4-one
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-3-yl]acetamide
1-(1-ethylpiperidin-4-yl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
3-[(5-ethyl-1,3,4-oxadiazol-2-yl)(methyl)amino]-1-phenylpropan-1-ol
9-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
3-(4-tert-butylbenzoyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(5-methyl-1,3-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
ethyl 2-[(5-{[(2S)-2-carbamoylpyrrolidin-1-yl]methyl}pyrimidin-2-yl)amino]acetate
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(pyridin-3-ylmethyl)oxolane-3-carboxamide
4-(1-{4-[2-(piperazin-1-ylmethyl)phenyl]phenyl}ethyl)morpholine
4-fluoro-N-{[4-(2-methylpropyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
2-{5-[2-(1H-imidazol-2-yl)phenyl]-1,2,4-oxadiazol-3-yl}pyrazine
(3S,4R)-1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
1-[(3-{[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-2-yl)piperazine
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
2-{4-[(2,5-dimethylphenyl)methyl]-1-(2,2-dimethylpropyl)piperazin-2-yl}ethan-1-ol
2-(cyclopropylamino)-N-(3-hydroxypropyl)-N-(naphthalen-1-ylmethyl)acetamide
[3-({1-[4-(piperidine-1-carbonyl)pyridin-2-yl]pyrrolidin-3-yl}methyl)phenyl]methanol
7-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-methyl-5-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-1H-1,3-benzodiazole
1-(4-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-{2-[4-(trifluoromethyl)phenyl]ethyl}-1,2-oxazole-3-carboxamide
2-[(3,5-difluorophenyl)methyl]-8-(3-methyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(4-methoxyphenyl)ethan-1-one
1-(3-chlorophenyl)-4-{1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-3-yl}piperazine
1-[2-(piperidin-1-yl)ethyl]-3-{2-[2-(pyridin-2-yl)ethyl]phenyl}urea
2-methoxy-5-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}methyl)benzoic acid
3-ethyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-(piperidin-1-yl)ethyl]amine
N-{3-[6-amino-5-cyano-4-(1,2-dimethyl-1H-imidazol-5-yl)pyridin-2-yl]phenyl}acetamide
1-(2,1,3-benzoxadiazol-5-ylmethyl)-2-methyl-1,4-diazepan-5-one
2-(2,5-dimethylphenoxy)-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}propanamide
(4S)-1-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
4-acetamido-2-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}benzamide