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3-[(3R,4S)-1-(3,6-dimethylpyrazin-2-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[(2R,4R,6S)-2-cyclohexyl-6-(3-fluoro-5-methylphenyl)oxan-4-yl]acetamide
2-{[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
4-methyl-2-(1-{4-[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}propyl)pyridine
N-cyclohexyl-5-(methoxymethyl)-N-(pyridin-4-ylmethyl)furan-2-carboxamide
(1S,5R)-6-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane
(3S,9aR)-3-benzyl-8-(naphthalene-2-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-methoxypyrazine
2-cyclopentyl-1-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-2-phenylethan-1-one
N-cyclopropyl-4-[3-(dimethylamino)phenyl]benzamide
N-[(3S,4R)-1-(2,3-dimethylquinoxaline-6-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
9-[(5-hydroxy-2-methoxyphenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-2-{[(2-propoxyphenyl)formamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}-2,3-dihydro-1H-isoindole
2-methyl-N-[3-(oxolan-3-yl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
N-[(4-phenyloxan-4-yl)methyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
N,N-dimethyl-5-{[4-(1-methylpiperidin-4-yl)piperazin-1-yl]methyl}pyrimidin-2-amine
2-(pyridine-3-carbonyl)-7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline
2-[(4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidin-5-yl)formamido]-N-(2-fluoro-4-methylphenyl)acetamide
5-{4-[(dimethylamino)methyl]phenyl}pyrazin-2-amine
1'-(2,6-dimethylpyrimidine-4-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-methyl-3-(pyrrolidine-1-carbonyl)-N-{[3-(trifluoromethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[(6-cyclopropylpyrimidin-4-yl)amino]-N-methylethane-1-sulfonamide
N-(2-methyl-1-{7-[3-(prop-2-en-1-yloxy)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)propanamide
1-methyl-4-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,4-dihydroquinoline-3-carboxamide
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]propanamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2,4-dimethyl-1,3-thiazole-5-carboxamide
1,9-dimethyl-4-(2-propyl-1,3-thiazole-4-carbonyl)-1,4,9-triazaspiro[5.5]undecane
4-{[(3-methoxyphenyl)methyl]amino}-5-methyl-N-(1,2-oxazol-3-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1-(4,6-dimethylquinazolin-2-yl)piperidine-4-carboxamide
(4aS,7aR)-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-(oxolan-2-ylmethoxy)ethan-1-one
2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-{[2-(trifluoromethoxy)phenyl]methyl}-1H-imidazole
methyl (2R,4S)-4-hydroxy-1-[5-(3-methoxyphenyl)furan-2-carbonyl]piperidine-2-carboxylate
4-{1-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-methylpropan-2-yl}morpholine
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-N-[3-(3-oxopiperazin-1-yl)propyl]acetamide
3,5-dimethoxy-N-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)methyl]benzamide
methyl 6-{[2-(2-hydroxyethyl)piperidin-1-yl]methyl}-3-[(2E)-3-phenylprop-2-enamido]thieno[2,3-b]pyridine-2-carboxylate
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methylpiperazine
N-[3-(dimethylamino)propyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}ethan-1-one
6-methyl-2-oxo-5-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,2-dihydropyridine-3-carbonitrile
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(pyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-tert-butyl-2-(4,5-dimethyl-2-oxo-2,3-dihydro-1,3-oxazol-3-yl)butanamide
N,N-diethyl-2-{4-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}acetamide
N-{2-methoxy-4-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]phenyl}butanamide