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1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(thiophen-3-yl)propan-1-one
1-(methoxymethyl)-N-[(3R,4S)-1-[(1-methyl-1H-imidazol-5-yl)methyl]-4-propylpyrrolidin-3-yl]cyclobutane-1-carboxamide
4-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-1-(propan-2-yl)-1H-pyrazole
1-(pyridin-2-ylmethyl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-1,4-diazepane
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-3-yl)ethan-1-one
3-{5-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-(2-methoxyethyl)-8-[(4-methoxyphenyl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methyl-N-({6-methyl-2-[methyl(1H-pyrazol-5-ylmethyl)amino]quinolin-3-yl}methyl)-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
N-benzyl-5-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}pyrimidin-2-amine
2-(3-methoxyphenyl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}azetidine
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)amine
1-(diethylamino)-3-{4-[(2,2-dimethylmorpholin-4-yl)methyl]-2-methoxyphenoxy}propan-2-ol
3-(3-fluorophenyl)-4-(2-phenylbenzoyl)piperazin-2-one
1-cyclohexyl-6-hydroxy-4-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1,4-diazepan-2-one
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methylcyclopropanecarbonyl)piperidine
2-(2-methoxyacetyl)-N-(2-phenoxyethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-4-(oxan-4-yl)piperazine
N-(2-methoxyethyl)-2-methyl-N-(pyridin-3-ylmethyl)-1,3-thiazole-4-carboxamide
1-{2-[(3-chloro-4-methylphenyl)carbamoyl]ethyl}-N-methylpyrrolidine-3-carboxamide
4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-N,N-dimethyl-5,6,7,8-tetrahydroquinazolin-2-amine
1-(2-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(2-chloro-3-methoxyphenyl)-2-cyclopropyl-1H-imidazole
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}({[5-(methoxymethyl)furan-2-yl]methyl})(pyridin-4-ylmethyl)amine
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-4-methyl-1,2,3-thiadiazole-5-carboxamide
N-({1-[(2-phenylphenyl)methyl]pyrrolidin-3-yl}methyl)acetamide
N-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
2-[(3,5-difluorophenyl)methyl]-8-(3-hydroxypropyl)-2,8-diazaspiro[4.5]decan-3-one
3-hydroxy-3-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-1-phenylpyrrolidin-2-one
1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propan-1-one
4-(1H-imidazol-1-yl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
3-(4-ethylpiperazine-1-carbonyl)-N-(oxolan-3-ylmethyl)benzene-1-sulfonamide
3-fluoro-N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)benzamide
1-(1-benzofuran-2-ylmethyl)-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-3-phenyl-1H-pyrazole-4-carboxamide
1-methyl-2-(1-{[4-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1H-imidazol-2-yl)-1H-imidazole
ethyl 4-[(4-methoxyphenyl)methyl]-1-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}piperidine-4-carboxylate
5-{4-[3-(trifluoromethyl)phenoxy]piperidine-1-carbonyl}pyrrolidin-2-one
N-({7-[(2,6-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-(3-fluorophenyl)acetamide
1-{1-[2-amino-6-(propan-2-yl)pyrimidine-4-carbonyl]piperidin-3-yl}pyrrolidin-2-one
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[3-(pyrrolidin-1-yl)propyl]amino}methyl)phenoxy]propan-2-ol
6-methoxy-1-methyl-2-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1H-indole
N-({8-[2-(naphthalen-2-yl)acetyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)pyridine-2-carboxamide
7-(cyclopropylmethyl)-2-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
3-benzyl-8-(2,2-dimethylpropyl)-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[4-({1-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)phenyl]acetamide
1-(2-chlorophenyl)-4-{3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propanoyl}piperazin-2-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(thiophene-2-carbonyl)pyrrolidin-3-yl]-1-methyl-1H-pyrrole-2-carboxamide
(2E)-1-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-(pyridin-2-yl)prop-2-en-1-one