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1-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-[(6-methoxypyridin-3-yl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
4-(1-ethyl-1H-1,2,4-triazol-5-yl)-7-hydroxy-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-amine
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanoic acid
N-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]thiophene-2-sulfonamide
4-(4-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}phenyl)-2-methylbutan-2-ol
6-[4-(2-methoxyphenoxy)piperidin-1-yl]pyridine-2-carboxylic acid
1-methanesulfonyl-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}pyrrolidine-2-carboxamide
2-(4-{2-amino-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}phenyl)-2-methylpropanenitrile
(1R,9aR)-1-({[(2-ethoxypyridin-3-yl)methyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
2-(2,4-dimethoxyphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
3-{2-tert-butylimidazo[1,2-a]pyrimidin-3-yl}pyridine
4-[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]piperazin-2-one
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-4-(morpholin-4-yl)butan-1-one
3-(3-chloro-2-methylphenyl)-1-[(4-hydroxyazepan-4-yl)methyl]urea
(1R,5R)-6-[4-(dimethylamino)benzoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-{2-amino-6-[(propan-2-yl)amino]pyrimidin-4-yl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-benzyl-1-methyl-5-(2-methyl-1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-{[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenol
1-benzyl-5-[(2,6-difluorophenyl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(2-propyl-1H-imidazol-1-yl)-N-(pyridin-3-yl)furan-2-carboxamide
5-[({1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]piperidin-4-yl}amino)methyl]pyrrolidin-2-one
3-(2-methoxyphenyl)-N-{2-[(3-methyl-1H-pyrazol-5-yl)methyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}propanamide
N-(3-ethoxy-2-hydroxypropyl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
8-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-[4-(6-methoxypyrimidin-4-yl)-1H-pyrazol-1-yl]acetamide
8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aS,7aR)-2-(4-chloro-3-methyl-1H-pyrazole-5-carbonyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyrrolidine-3-carboxamide
2-(4-amino-1H-pyrazol-1-yl)-N-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]acetamide
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-benzyl-N-ethylpropanamide
dimethyl[(4-methyl-5-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
methyl 2-[(2,3-dihydro-1H-inden-5-yl)sulfamoyl]-6-(1-methylcyclopropanecarbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(methylamino)-N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]-1,3-thiazole-4-carboxamide
2-[4-(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1H-imidazol-2-yl)phenoxy]ethan-1-ol
4-{4-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]piperidin-1-yl}-6-methyl-2-(propan-2-yl)pyrimidine
2-(4-ethoxyphenyl)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-2-(3-phenyl-1H-pyrazol-1-yl)acetamide
2-{1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidin-2-yl}-1H-1,3-benzodiazole
(3S,4S)-4-cyclopropyl-1-[2-(2-fluorophenyl)acetyl]pyrrolidine-3-carboxylic acid
5-[3-(naphthalene-1-carbonyl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-methyl-3-(5-methylfuran-2-yl)-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-1H-pyrazole-5-carboxamide
N-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N-methylpyridine-2-carboxamide
1-(oxolane-3-carbonyl)-4-(pyridin-3-yl)piperazine
2-[(6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}quinazolin-4-yl)amino]ethan-1-ol
1-(4-methylbenzenesulfonyl)-4-(oxane-2-carbonyl)piperazine
1-[4-(4,6-dimethoxypyrimidin-2-yl)-6-hydroxy-1,4-diazepan-1-yl]ethan-1-one
1-(adamantan-1-yl)-4-(4-methyl-1,3-oxazole-5-carbonyl)piperazine