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5-{[(2,5-difluorophenyl)methyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{[4-methyl-5-({[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
1-({2-methyl-7-[(1-propyl-1H-imidazol-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)propan-2-ol
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(4aS,8aR)-6-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
1-methyl-5-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
5-(hydroxymethyl)-N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-propylpyrrolidin-3-yl]furan-2-carboxamide
6-methyl-2-propyl-N-[2-(1H-1,2,4-triazol-1-yl)propyl]pyrimidin-4-amine
N-(2-fluoro-5-methylphenyl)-N'-{3-[(pyridin-3-yl)amino]propyl}butanediamide
3-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}propan-1-ol
1-[4-chloro-3-(trifluoromethyl)phenyl]-4-(5-methyl-1,3-oxazole-4-carbonyl)piperazine
ethyl 1-(1H-1,3-benzodiazole-5-carbonyl)-3-(2-phenoxyethyl)piperidine-3-carboxylate
4-(2,6-dimethylpyridin-3-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidin-2-amine
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-[(2,3,6-trifluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
N5-[(1-ethylpiperidin-3-yl)methyl]-N6-(2-methoxyethyl)-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-butyl-4-[(3-methylphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-({1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,3-thiazol-4-ylmethyl)amine
N-(1,4-dioxan-2-ylmethyl)-N,6-dimethyl-2-phenylpyrimidin-4-amine
4-methyl-2-(propan-2-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]-1,3-thiazole-5-carboxamide
8-[(2,5-difluorophenyl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
7-(1,3-benzothiazol-2-yl)-4-(oxane-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4,6-dimethylpyrimidin-2-amine
4-{4-[(4-methylphenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylpropyl)-N-(propan-2-yl)acetamide
N-(1-{4-[(1E)-pent-1-en-1-yl]phenyl}ethyl)acetamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
N-[(3S,4R)-1-(2,5-dimethylfuran-3-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
N-[(2-ethoxyphenyl)methyl]-4-hydroxy-N-methyl-2-(4-methylphenyl)pyrimidine-5-carboxamide
8-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
3-(3-methoxypropyl)-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
1-{2-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}azepan-2-one
1-[4-(pyrrolidin-1-yl)pentanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-methyl-1-[3-(pyridin-3-yl)propanoyl]piperidine-3-carbonitrile
[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl](pyridin-2-yl)methanol
2-[5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl]-2-azabicyclo[2.2.1]hept-5-ene
N-{1-[2-(2-ethylpiperidin-1-yl)-2-oxoethyl]-1H-pyrazol-4-yl}-3-phenoxypropanamide
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetamide
2-[(2,1,3-benzoxadiazol-4-ylmethyl)(pyridin-3-ylmethyl)amino]butan-1-ol
5-[2-(2-ethoxyphenoxy)ethyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine
4-(5-fluoro-2-methylbenzenesulfonyl)-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N2-[2-(dimethylamino)ethyl]-N5-(3-methylphenyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2,5-dicarboxamide
(5-{[8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}furan-2-yl)methanol
3-amino-1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
N-[2-(benzylsulfanyl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-{[3-(2-methoxypyridin-3-yl)phenyl]methyl}acetamide
1-[1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)azetidin-3-yl]piperidine
N,N-dimethyl-5-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1,9-dioxaspiro[5.5]undecan-4-amine