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8-[(3-hydroxyphenyl)methyl]-1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[4-(2-chlorophenoxy)piperidin-1-yl]-2-[methyl(piperidin-4-yl)amino]ethan-1-one
{3-[(3-chlorophenyl)methyl]-1-[(2,6-dimethoxyphenyl)methyl]piperidin-3-yl}methanol
1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
3-(2-fluoropyridin-3-yl)-1-[1-(pyrazin-2-yl)piperidin-3-yl]urea
methyl 5-[3-(2-fluorophenyl)pyrrolidin-1-yl]-5-oxopentanoate
1-methyl-3-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-1-[1-(4-methylpyridin-2-yl)propan-2-yl]urea
N-{1-[(2-ethylpyrimidin-4-yl)methyl]pyrrolidin-3-yl}acetamide
2-(2,3-difluoro-4-methoxyphenyl)-1H-1,3-benzodiazole-5-carbonitrile
1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
(2R)-2-[5-(4-methyl-2-oxo-2H-chromen-7-yl)-4-phenyl-1H-imidazol-1-yl]propanamide
2-methyl-5-(4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
3-(1-methyl-1H-pyrazol-4-yl)-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)propanamide
1-({6-[4-(benzyloxy)-2-methylphenyl]pyridin-3-yl}methyl)-4-methylpiperazine
4-{2-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-1H-imidazol-1-yl}-1-(4-methylphenyl)pyrrolidin-2-one
2-(5-{1-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine
4-{4-[3-(methoxymethyl)piperidin-1-yl]piperidin-1-yl}-N-[2-(morpholin-4-yl)ethyl]benzamide
4-benzyl-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-ethyl-2-{4-[6-(1-hydroxyethyl)pyridin-2-yl]piperazin-1-yl}acetamide
(2R,6R)-4-[2-(cyclohexylcarbamoyl)ethyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{1-[1-(oxan-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
(2R,6S)-4-(1-{1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carbonyl}piperidin-4-yl)-2,6-dimethylmorpholine
1-methyl-3,8-bis(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[3-(1H-pyrazol-1-yl)propyl](pyridin-4-ylmethyl)amine
1-cyclohexyl-3-(cyclopropylmethyl)-5-(4-methylpiperazine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-(2-{6-[(2-methoxyethyl)carbamoyl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-yl}acetamido)-2-methylpropanoic acid
6-[3-(1,3-benzoxazol-2-yl)piperidine-1-carbonyl]-2-cyclohexyl-1,3-benzoxazole
N-(3,5-dimethoxyphenyl)-3-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-3-yl)propanamide
(1R,5R)-3-cyclobutanecarbonyl-6-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(2-{6-oxa-9-azaspiro[4.5]decan-9-yl}pyrimidin-4-yl)piperidin-3-ol
2-(adamantan-1-yl)-5-[3-(aminomethyl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
3-({5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)propane-1,2-diol
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-(4-hydroxyphenyl)benzamide
4-(5-{[(5-chloropyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)-1-methyl-2-phenylpiperazine
7-fluoro-3-methyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1-benzofuran-2-carboxamide
1-[(5-chlorofuran-2-yl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
2-[(2S)-3-phenyl-2-{[5-(propan-2-yl)-1,2-oxazol-3-yl]formamido}propanamido]acetic acid
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylazepane-2-carboxamide
1-(3,5-difluorophenyl)-N-(quinolin-5-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-(pyridin-2-ylmethyl)-2-{4-[4-({2-[4-(trifluoromethyl)phenyl]ethyl}amino)piperidin-1-yl]phenyl}acetamide
1-methyl-4-(3-methyl-5-{2-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-1,2,4-triazol-1-yl)piperidine
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-phenyl-3-(pyridin-2-yl)propanamide
1-{4-[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-3-methyl-2-phenoxybutan-1-one
3-chloro-N-cyclopentyl-4-({1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}oxy)benzamide
1-{2-[2-(3-chloro-2,6-difluorophenyl)-1H-imidazol-1-yl]ethyl}piperidine
N-methyl-5-(morpholin-4-ylmethyl)-N-(pyridin-2-ylmethyl)-1,2-oxazole-3-carboxamide
N,N,4,5-tetramethyl-6-(1H-pyrazol-3-yl)pyrimidin-2-amine
2-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)amino)methyl]phenol
4-{[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]methyl}-2,6-dimethoxyphenol
2-[2-(3-methoxypiperidin-1-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid